4- (HETEROCYCLYL- FUSED PHENYL)- 3- (PHENYL OR PYRID -2- YL) PYRAZOLES AS INHIBITORS OF THE ALK-5- RECEPTOR - Patent 1656367

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EP 1 656 367 A1

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(43)	Date of publication:
	17.05.2006 Bulletin 2006/20

(21)	Application number: 04739898.7

(22)	Date of filing: 14.06.2004

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International Patent Classification (IPC):

C07D 401/14^(1990.01)
A61K 31/538^(2000.01)

C07D 413/14^(1990.01)
A61P 13/12^(2000.01)

(86)	International application number:
	PCT/EP2004/006427

(87)	International publication number:
	WO 2004/111036 (23.12.2004 Gazette 2004/52)

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
	Designated Extension States:
	HR LT LV

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Priority:

16.06.2003 GB 0313915

(71)	Applicant: SMITHKLINE BEECHAM CORPORATION
	Philadelphia, Pennsylvania 19101 (US)

(72)	Inventors:
	DODIC, Nerina, Laboratoire GlaxoSmithKline F-91951 Les Ulis (FR) DONCHE, Frederic, Laboratoire GlaxoSmithKline F-91951 Les Ulis (FR) GELLIBERT, Francoise Jeanne, Lab. GlaxoSmithKline F-91951 Les Ulis (FR)

(74)	Representative: Sardharwala, Fatema Elyasali
	GlaxoSmithKline Corporate Intellectual Property 980 Great West Road GB-Brentford, Middlesex TW8 9GS GB-Brentford, Middlesex TW8 9GS (GB)

(54)	4- (HETEROCYCLYL- FUSED PHENYL)- 3- (PHENYL OR PYRID -2- YL) PYRAZOLES AS INHIBITORS OF THE ALK-5- RECEPTOR