(19)
(11) EP 1 687 268 A1

(12)

(43) Date of publication:
09.08.2006 Bulletin 2006/32

(21) Application number: 04810567.0

(22) Date of filing: 08.11.2004
(51) International Patent Classification (IPC): 
C07D 207/14(2006.01)
C07D 213/53(2006.01)
C07D 211/62(2006.01)
C07D 211/52(2006.01)
C07D 211/42(2006.01)
C07D 211/66(2006.01)
C07D 211/44(2006.01)
C07D 471/10(2006.01)
C07D 207/08(2006.01)
C07D 403/12(2006.01)
C07D 211/58(2006.01)
C07D 211/46(2006.01)
C07D 213/82(2006.01)
C07D 401/12(2006.01)
C07D 211/38(2006.01)
(86) International application number:
PCT/US2004/037258
(87) International publication number:
WO 2005/047249 (26.05.2005 Gazette 2005/21)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LU MC NL PL PT RO SE SI SK TR

(30) Priority: 10.11.2003 US 519002 P

(71) Applicant: Schering Aktiengesellschaft
13353 Berlin (DE)

(72) Inventors:
  • DAVEY, David
    El Sobrante, CA 94803 (US)
  • LEE, Wheeseong
    Orinda, CA 94563 (US)
  • LU, Shou-Fu
    San Ramon, CA 94583 (US)
  • PHILLIPS, Gary
    Pleasant Hill, CA 94523 (US)
  • WEI, Guo, Ping
    San Ramon, CA 94582 (US)
  • YE, Bin
    Moraga, CA 94556 (US)

(74) Representative: Pohlman, Sandra M. et al
Dörries Frank-Molnia & Pohlman, Triftstrasse 13
80538 München
80538 München (DE)

   


(54) BENZYLETHER AMINE COMPOUNDS USEFUL AS CCR-5 ANTAGONISTS