(19)
(11) EP 1 740 557 A1

(12)

(43) Date of publication:
10.01.2007 Bulletin 2007/02

(21) Application number: 05716548.2

(22) Date of filing: 07.04.2005
(51) International Patent Classification (IPC): 
C07D 265/36(2006.01)
A61K 31/538(2006.01)
 C07D 215/227(2006.01)
A61P 13/02(2006.01)
(86) International application number:
PCT/EP2005/003632
(87) International publication number:
WO 2005/103018 (03.11.2005 Gazette 2005/44)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR

(30) Priority: 20.04.2004 EP 04009274

(71) Applicant: Bayer HealthCare AG
51368 Leverkusen (DE)

(72) Inventors:
  • FUJISHIMA, Hiroshi
    Nara-shi, Nara 631-0801 (JP)
  • MOGI, Muneto
    4058 Basel (CH)
  • YUASA, Hiroaki
    Itano-gunn, Tokushima-ken, 771-0205 (JP)
  • TAIJIMI, Masaomi
    Canterbury, Kent CT1 3BZ (GB)
  • YAMAMOTO, Noriyuki
    Osaka-fu, Osaka 577-0013 (JP)
  • HAYASHI, Fumihiko
    Soraku-gun, Kyoto 619-0224 (JP)
  • TSUKIMI, Yasuhiro
    Hyogo 661-0975 (JP)
  • GUPTA, Jang
    40489 Düsseldorf (DE)

   


(54) UREA DERIVATIVES AS ANTAGONISTS OF THE VANILLOID RECEPTOR (VR1)