(19)
(11) EP 1 771 416 A1

(12)

(43) Date of publication:
11.04.2007 Bulletin 2007/15

(21) Application number: 04806738.3

(22) Date of filing: 28.07.2004
(51) International Patent Classification (IPC): 
C07D 211/32(2006.01)
A61P 25/28(2006.01)
A61K 31/445(2006.01)
(86) International application number:
PCT/IN2004/000227
(87) International publication number:
WO 2006/011154 (02.02.2006 Gazette 2006/05)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
Designated Extension States:
AL HR LT LV

(71) Applicant: USV Limited
Mumbai 400088, Maharashtra (IN)

(72) Inventors:
  • TARUR, Venkatasubramanian Radhakrishnan
    Mumbai 400 080, Maharashtra (IN)
  • SATHE, Dhananjay Govind
    Thane 400 602, Maharashtra (IN)
  • NAIDU, Avinash Venkataraman
    Vishnu Nagar, Dombivli 421 202 (IN)
  • AHER, Umesh Parashram
    Kalyan 421 301, Maharashtra (IN)
  • SAWANT, Kamlesh Digambar
    Mumbai 400 030, Maharashtra (IN)

(74) Representative: Henkel, Feiler & Hänzel 
Patentanwälte Maximiliansplatz 21
80333 München
80333 München (DE)

   


(54) A NOVEL POLYMORPH OF (1-BENZYL-4-[(5,6-DIMETHOXY-1-INDANONE)-2-YL] METHYL PIPERIDINE HYDROCHLORIDE (DONEPEZIL HYDROCHLORIDE) AND A PROCESS FOR PRODUCING THEREOF