(19)
(11) EP 1 771 431 A1

(12)

(43) Date of publication:
11.04.2007 Bulletin 2007/15

(21) Application number: 05760356.5

(22) Date of filing: 03.06.2005
(51) International Patent Classification (IPC): 
C07D 307/28(2006.01)
(86) International application number:
PCT/US2005/019669
(87) International publication number:
WO 2005/118565 (15.12.2005 Gazette 2005/50)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR
Designated Extension States:
AL BA HR LV MK YU

(30) Priority: 03.06.2004 US 576642 P
10.11.2004 US 626769 P
18.03.2005 US 663300 P

(71) Applicant: Eisai Co., Ltd.
Tokyo 112-8088 (JP)

(72) Inventors:
  • AUSTAD, Brian
    Tewksbury, MA 01876 (US)
  • CHASE, Charles, E.
    Londonderry, NH 03053 (US)
  • FANG, Francis, G.
    Andover, MA 01810 (US)

(74) Representative: Sexton, Jane Helen 
J.A. KEMP & CO. 14 South Square Gray's Inn
London WC1R 5JJ
London WC1R 5JJ (GB)

   


(54) INTERMEDIATES FOR THE PREPARATION OF HALICHONDRIN B