(19)
(11) EP 1 773 398 A2

(12)

(88) Date of publication A3:
30.03.2006

(43) Date of publication:
18.04.2007 Bulletin 2007/16

(21) Application number: 05788746.5

(22) Date of filing: 09.06.2005
(51) International Patent Classification (IPC): 
A61K 47/00(2006.01)
A61K 31/42(2006.01)
C07D 239/02(2006.01)
C07D 211/84(2006.01)
C07C 303/00(2006.01)
A61K 31/40(2006.01)
A61K 31/505(2006.01)
C07D 261/04(2006.01)
C07D 209/12(2006.01)
(86) International application number:
PCT/US2005/020770
(87) International publication number:
WO 2005/120515 (22.12.2005 Gazette 2005/51)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR

(30) Priority: 10.06.2004 WO PCT/US2004/018502
10.06.2004 US 865743
09.12.2004 US 635019 P

(71) Applicant: Kalypsys, Inc.
San Diego, CA 92121 (US)

(72) Inventors:
  • MALECHA, James
    San Diego, California 92130 (US)
  • NOBLE, Stewart
    San Diego, California 92130 (US)
  • HASSIG, Christian
    San Diego, California 92126 (US)
  • WASH, Paul
    San Diego, California 92103 (US)
  • WILEY, Brandon
    Encinitas, California 92024 (US)
  • LAWRENCE, Charles
    San Diego, California 92104 (US)
  • HOFFMAN, Timothy
    San Diego, California 92126 (US)

(74) Representative: Albrecht, Thomas 
Kraus & Weisert Patent- und Rechtsanwälte Thomas-Wimmer-Ring 15
80539 München
80539 München (DE)

   


(54) NOVEL SULFONAMIDES AS INHIBITORS OF HISTONE DEACETYLASE FOR THE TREATMENT OF DISEASE