(19)
(11) EP 1 793 806 A2

(12)

(88) Date of publication A3:
27.07.2006

(43) Date of publication:
13.06.2007 Bulletin 2007/24

(21) Application number: 05803721.9

(22) Date of filing: 29.09.2005
(51) International Patent Classification (IPC): 
A61K 9/14(2006.01)
A61K 9/20(2006.01)
A61K 9/50(2006.01)
A61K 9/16(2006.01)
A61K 9/48(2006.01)
(86) International application number:
PCT/US2005/034587
(87) International publication number:
WO 2006/039268 (13.04.2006 Gazette 2006/15)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

(30) Priority: 30.09.2004 US 614891 P

(71) Applicant: EASTMAN CHEMICAL COMPANY
Kingsport, TN 37660 (US)

(72) Inventors:
  • HYATT, John, Anthony
    Kingsport, TN 37664 (US)
  • ZIMA, George, Chester
    Kingsport, TN 37660 (US)
  • EDGAR, Kevin, Joseph
    Kingsport, TN 37663 (US)
  • NAVARRO, Lisa, Tonner
    High Point, NC 27261 (US)
  • LEHR, Claus-Michael
    66125 Saarbrucken-Dudweiler (DE)
  • COLLNOT, Eva-Maria
    66564 Ottweiler (DE)
  • SINGLETON, Andy, Hugh
    Kingsport, TN 37664 (US)
  • BALDES, Christiane
    66123 Saarbrucken (DE)
  • SCHAFER, Ulrich, Friedrich
    66280 Sulzbach (DE)
  • WEMPE, Michael, Fitzpatrick
    Kingsport, TN 37660 (US)

(74) Representative: Rees, Kerry et al
FJ Cleveland 40-43 Chancery Lane
London WC2A 1JQ
London WC2A 1JQ (GB)

   


(54) PHARMACEUTICAL FORMULATIONS CONTAINING VITAMIN E TPGS MOLECULES THAT SOLUBILIZE LIPOPHILIC DRUGS WITHOUT SIGNIFICANT EFFLUX INHIBITION, AND USE OF SUCH FORMULATIONS