<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.0//EN" "ep-patent-document-v1-0.dtd"><ep-patent-document id="EP05805719A1" file="05805719.1" lang="en" country="EP" doc-number="1793843" kind="A1" date-publ="20070613" status="n" dtd-version="ep-patent-document-v1-1"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIRO..CY..TRBGCZEEHUPLSK....IS..........</B001EP><B003EP>*</B003EP><B005EP>X</B005EP><B007EP>DIM360 (Ver 1.5  21 Nov 2005) -  1100000/0 1710000/0</B007EP></eptags></B000><B100><B110>1793843</B110><B130>A1</B130><B140><date>20070613</date></B140><B190>EP</B190></B100><B200><B210>05805719.1</B210><B220><date>20050930</date></B220><B240><B241><date>20070328</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>614800 P</B310><B320><date>20040930</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20070613</date><bnum>200724</bnum></B405><B430><date>20070613</date><bnum>200724</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>A61K  38/12        20060101AFI20060822BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/675       20060101ALI20060822BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07F   9/553       20060101ALI20060822BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07K   5/12        20060101ALI20060822BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61P  35/00        20060101ALI20060822BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>MAKROZYKLISCHE SH2-DOMÄNE BINDENDE INHIBITOREN</B542><B541>en</B541><B542>MACROCYCLIC SH2 DOMAIN BINDING INHIBITORS</B542><B541>fr</B541><B542>INHIBITEURS DE LIAISON DE DOMAINE SH2 MACROCYCLIQUE</B542></B540></B500><B700><B710><B711><snm>Government of the United States of America, 
Represented by the Secretary, Department 
of Health and Human Services</snm><iid>07886010</iid><irf>MK-P35264EPPC</irf><adr><str>Office of Technology Transfer 
6011 Executive Boulevard, Suite 325</str><city>Rockville, Maryland 20852</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>BURKE, JR., Terrence R.</snm><adr><str>7400 Lakeview Dr. , No.410</str><city>Bethesda MD 20817</city><ctry>US</ctry></adr></B721><B721><snm>SHI, Zhen-Dan</snm><adr><str>8506 Bradmoor Drive</str><city>Bethesda MD 20817</city><ctry>US</ctry></adr></B721><B721><snm>OISHI, Shinya</snm><adr><str>50-313 Higashitakeya-machi, Sakyo-ku.</str><city>Kyoto 606-8393</city><ctry>JP</ctry></adr></B721><B721><snm>LIU, Fa</snm><adr><str>313 Selwyn Drive, Apt. 2D</str><city>Frederick, MD 21701</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Hoechst, Bruno Werner</snm><sfx>et al</sfx><iid>09224521</iid><adr><str>Bohest Intellectual Property 
A. Braun Braun Héritier Eschmann AG 
Holbeinstrasse 36-38</str><city>4051 Basel</city><ctry>CH</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>US2005035246</anum></dnum><date>20050930</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2006039527</pnum></dnum><date>20060413</date><bnum>200615</bnum></B871></B870></B800></SDOBI></ep-patent-document>