(19)

(11)

EP 1 794 177 A2

(12)

(88) Date of publication A3: 17.08.2006 (43) Date of publication: 13.06.2007 Bulletin 2007/24 (21) Application number: 05805074.1 (22) Date of filing: 25.08.2005

(51) International Patent Classification (IPC):  C07J 53/00(2006.01) C07J 21/00(2006.01) (86) International application number: PCT/IB2005/002757 (87) International publication number: WO 2006/032970 (30.03.2006 Gazette 2006/13)

(84) Designated Contracting States: AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR (30) Priority: 09.09.2004 US 608425 P 22.09.2004 US 612133 P (71) Applicant: Pharmacia Corporation Peapack, NJ 07977 (US)

(72) Inventors: ABBAS, Zaheer Chesterfield, MO 63017-1732 (US) BAUER, Michael Chesterfield, MO 63017-1732 (US) CARLOS, Marlon V. Chesterfield, MO 63017-1732 (US) DAVID, Paul Chesterfield, MO 63017-1732 (US) FRANZYK, Thaddeus Chesterfield, MO 63017-1732 (US) KIM, Chung C. Chesterfield, MO 63017-1732 (US) LAWSON, Jon P. Chesterfield, MO 63017-1732 (US) MAISTO, Keith D. Chesterfield, MO 63017-1732 (US) McKENZIE, David Chesterfield, MO 63017-1732 (US) POZZO, Mark Chesterfield, MO 63017-1732 (US) WIECZOREK, Joseph Chesterfield, MO 63017-1732 (US) (74) Representative: Kingsbury, Oliver William et al Pfizer Limited European Patent Department IPC 748 GB-Sandwich, Kent CT13 9NJ GB-Sandwich, Kent CT13 9NJ (GB)