(19)

(11)

EP 1 809 245 A2

(12)

(88) Date of publication A3: 04.08.2005 (43) Date of publication: 25.07.2007 Bulletin 2007/30 (21) Application number: 04817762.0 (22) Date of filing: 09.09.2004

(51) International Patent Classification (IPC):  A61K 9/127(2006.01) (86) International application number: PCT/US2004/029265 (87) International publication number: WO 2005/053605 (16.06.2005 Gazette 2005/24)

(84) Designated Contracting States: AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR (30) Priority: 09.09.2004 US 501816 P 09.09.2003 US 501818 P (71) Applicant: GILEAD SCIENCES, INC. Foster City, CA 94404 (US)	(72) Inventors: JENSEN, Gerard Brea, CA 92821 (US) HU, Ning San Gabriel, CA 91775 (US) PETRASEK, Danny Los Angeles, CA 90047 (US) (74) Representative: Reitstötter - Kinzebach  Patentanwälte, Sternwartstrasse 4 81679 München 81679 München (DE)