<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.0//EN" "ep-patent-document-v1-0.dtd"><ep-patent-document id="EP05712354A1" file="05712354.9" lang="en" country="EP" doc-number="1848273" kind="A1" date-publ="20071031" status="n" dtd-version="ep-patent-document-v1-1"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSKBAHRISYU........</B001EP><B003EP>*</B003EP><B005EP>X</B005EP><B007EP>DIM360 (Ver 1.5  21 Nov 2005) -  1100000/0 1710000/0</B007EP></eptags></B000><B100><B110>1848273</B110><B130>A1</B130><B140><date>20071031</date></B140><B190>EP</B190></B100><B200><B210>05712354.9</B210><B220><date>20050131</date></B220><B240><B241><date>20070831</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B400><B405><date>20071031</date><bnum>200744</bnum></B405><B430><date>20071031</date><bnum>200744</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>A01N  43/04        20060101AFI20060822BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/70        20060101ALI20060822BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>18-GLIEDRIGE MAKROCYCLEN UND IHRE ANALOGA</B542><B541>en</B541><B542>18-MEMBERED MACROCYCLES AND ANALOGS THEREOF</B542><B541>fr</B541><B542>MACROCYCLES A 18 CHAINONS ET LEURS ANALOGUES</B542></B540></B500><B700><B710><B711><snm>Optimer Pharmaceuticals, Inc.</snm><iid>04693830</iid><irf>MORCM/P38620EP</irf><adr><str>10110 Sorrento Valley Road, 
Suite C</str><city>San Diego, CA 92121</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>SHUE, Youe-Kong</snm><adr><str>7869 Via Teca</str><city>Carlsbad, CA 92009</city><ctry>US</ctry></adr></B721><B721><snm>HWANG, Chan-Kou</snm><adr><str>11402 Ocean Ridge Way</str><city>San Diego, CA 92130</city><ctry>US</ctry></adr></B721><B721><snm>CHIU, Yu-Hung</snm><adr><str>13993 Recuerdo Drive</str><city>Del Mar, CA 92014</city><ctry>US</ctry></adr></B721><B721><snm>ROMERO, Alex</snm><adr><str>2219 Howard Avenue</str><city>San Diego, CA 92104</city><ctry>US</ctry></adr></B721><B721><snm>BABAKHANI, Farah</snm><adr><str>10955 Elderwood Road</str><city>San Diego, CA 92131</city><ctry>US</ctry></adr></B721><B721><snm>SEARS, Pamela</snm><adr><str>11883 Spruce Run Drive C</str><city>San Diego, CA 92131</city><ctry>US</ctry></adr></B721><B721><snm>OKUMU, Franklin</snm><adr><str>3649 Victor Avenue</str><city>Oakland, CA 94619</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Stevens, Ian Edward</snm><iid>00078682</iid><adr><str>Eric Potter Clarkson LLP 
Park View House 
58 The Ropewalk</str><city>Nottingham NG1 5DD</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B844EP><B845EP><ctry>AL</ctry><date>20070831</date></B845EP><B845EP><ctry>BA</ctry><date>20070831</date></B845EP><B845EP><ctry>HR</ctry><date>20070831</date></B845EP><B845EP><ctry>LV</ctry><date>20070831</date></B845EP><B845EP><ctry>MK</ctry><date>20070831</date></B845EP><B845EP><ctry>YU</ctry><date>20070831</date></B845EP></B844EP><B860><B861><dnum><anum>US2005002887</anum></dnum><date>20050131</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2006085838</pnum></dnum><date>20060817</date><bnum>200633</bnum></B871></B870></B800></SDOBI></ep-patent-document>