(19)
(11) EP 1 865 775 A1

(12)

(43) Date of publication:
19.12.2007 Bulletin 2007/51

(21) Application number: 06749458.3

(22) Date of filing: 06.04.2006
(51) International Patent Classification (IPC): 
A01N 43/58(2006.01)
A01N 43/54(2006.01)
A61K 31/50(2006.01)
A61K 31/517(2006.01)
C07D 237/30(2006.01)
C07D 401/00(2006.01)
C07D 413/00(2006.01)
C07D 419/00(2006.01)
C07D 217/22(2006.01)
A01N 43/60(2006.01)
A01N 43/42(2006.01)
A61K 31/495(2006.01)
A61K 31/47(2006.01)
C07D 239/72(2006.01)
C07D 403/00(2006.01)
C07D 417/00(2006.01)
C07D 217/00(2006.01)
(86) International application number:
PCT/US2006/012915
(87) International publication number:
WO 2006/108107 (12.10.2006 Gazette 2006/41)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

(30) Priority: 06.04.2005 US 669030 P

(71) Applicant: IRM, LLC
Hamilton, HM LX (BM)

(72) Inventors:
  • MICHELLYS, Pierre-Yves
    San Marcos, California 92069 (US)
  • WEN, Ke
    Shanghai 201101 (CN)
  • PETRASSI, Michael, H.
    Cardiff, California 92007 (US)
  • PEI, Wei
    San Diego, California 92126 (US)

(74) Representative: Kiddle, Simon John 
Mewburn Ellis LLP York House, 23 Kingsway
London WC2B 6HP
London WC2B 6HP (GB)

   


(54) DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF STEROID HORMONE NUCLEAR RECEPTORS