(19)
(11) EP 1 942 105 B8

(12) CORRECTED EUROPEAN PATENT SPECIFICATION
Note: Bibliography reflects the latest situation

(15) Correction information:
Corrected version no 1 (W1 B1)

(48) Corrigendum issued on:
13.08.2014 Bulletin 2014/33

(45) Mention of the grant of the patent:
16.04.2014 Bulletin 2014/16

(21) Application number: 06822035.9

(22) Date of filing: 23.10.2006
(51) International Patent Classification (IPC): 
C07D 239/14(2006.01)
A61K 31/505(2006.01)
A61K 31/535(2006.01)
A61K 31/541(2006.01)
A61K 31/55(2006.01)
A61K 31/554(2006.01)
A61P 43/00(2006.01)
C07D 265/08(2006.01)
C07D 279/06(2006.01)
C07D 281/02(2006.01)
A61K 31/426(2006.01)
A61K 31/506(2006.01)
A61K 31/54(2006.01)
A61K 31/5415(2006.01)
A61K 31/551(2006.01)
A61P 25/28(2006.01)
C07D 239/24(2006.01)
C07D 277/18(2006.01)
C07D 279/08(2006.01)
C07D 405/04(2006.01)
(86) International application number:
PCT/JP2006/321015
(87) International publication number:
WO 2007/049532 (03.05.2007 Gazette 2007/18)

(54)

AMINODIHYDROTHIAZINE DERIVATIVE

AMINODIHYDROTHIAZIN-DERIVAT

DERIVE AMINODIHYDROTHIAZINE


(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

(30) Priority: 25.10.2005 JP 2005309642
20.03.2006 JP 2006076636

(43) Date of publication of application:
09.07.2008 Bulletin 2008/28

(60) Divisional application:
13150548.9 / 2612854
13150550.5 / 2597087

(73) Proprietor: Shionogi & Co., Ltd.
Osaka 541-0045 (JP)

(72) Inventors:
  • KOBAYASHI, Naotake
    Osaka-shi, Osaka 5530002 (JP)
  • UEDA, Kazuo
    Osaka-shi, Osaka 5530002 (JP)
  • ITOH, Naohiro
    Koka-shi Shiga 5203423 (JP)
  • SUZUKI, Shinji
    Osaka-shi, Osaka 5530002 (JP)
  • SAKAGUCHI, Gaku
    Koka-shi Shiga 5203423 (JP)
  • KATO, Akira
    Koka-shi Shiga 5203423 (JP)
  • YUKIMASA, Akira
    Osaka-shi, Osaka 5530002 (JP)
  • HORI, Akihiro
    Osaka-shi, Osaka 5530002 (JP)
  • KORIYAMA, Yuji
    Osaka-shi, Osaka 5530002 (JP)
  • HARAGUCHI, Hidekazu
    Osaka-shi, Osaka 5530002 (JP)
  • YASUI, Ken
    Osaka-shi, Osaka 5530002 (JP)
  • KANDA, Yasuhiko
    Osaka-shi, Osaka 5530002 (JP)

(74) Representative: Vossius & Partner 
Siebertstrasse 4
81675 München
81675 München (DE)


(56) References cited: : 
EP-A1- 0 713 704
WO-A1-2004/014843
WO-A2-2005/111031
JP-A- 08 231 521
JP-A- 2005 509 651
JP-A- 2005 526 005
US-A1- 2005 165 080
WO-A1-02/096897
WO-A1-2004/043916
CH-A- 484 184
JP-A- 2004 149 429
JP-A- 2005 517 634
JP-A- 2005 531 520
   
  • SCHUBERT ET AL.: "Neue Synthesen von 2-Amino-5,6-dihydro-4H-1,3-thiazinen", ARCHIV DER PHARMAZIE, vol. 301, no. 10, 1968, pages 750-762, XP002632395,
  • LIEBSCHER J. ET AL.: '2-ARYLIMINO-3-THIAZOLINES - FORMATION OF UNUSUAL TAUTOMERS OF 2-ARYLAMINO-THIAZOLINES - A REVISION' TETRAHEDRON LETTERS vol. 26, no. 35, 1985, pages 4179 - 4180, XP003011652
  • GARCIA FERNANDEZ J.M. ET AL.: 'Syntheses and Spectral Properties of beta-Idoureas and 2-Amino-4,4-diphenyl-2-oxazolines' JOURNAL OF HETEROCYCLIC CHEMISTRY vol. 28, no. 3, 1991, pages 777 - 780, XP003011653
  • SCHAUMANN. ET AL.: 'Stickstoffhaltige Funfring-Heterocyclen aus Carbodiimiden oder Ketenimine mit 3-Dimethylamino-2H-azirinen' LIEBIGS ANNALEN DER CHEMIE no. 2, 1981, pages 290 - 305, XP003011654
  • GARCIA FERNANDEZ J.M. ET AL.: 'Syntheses of beta-iodourea derivatives of carbohydrates and glycosylamino-oxazolines' CARBOHYDRATE RESEARCH vol. 216, 1991, pages 21 - 32, XP003011655
  • COHEN N. ET AL.: 'Synthesis of 2-Amino-5-, 6-dihydro-4H-1,3-thiazines and Related Compounds by Acid Catalyzed Cyclization of Allylic Isothiuronium Salts' JOURNAL OF HETEROCYCLIC CHEMISTRY vol. 14, no. 5, 1977, pages 717 - 723, XP003011656
  • CAMBIE R.C. ET AL.: 'vic-Iodothiocyanates and Iodoisothiocyanates. Part 2. New Syntheses of Thiazolidin-2-ones and 2-Amino-2-thiazolines' JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS I no. 3, 1979, pages 765 - 770, XP003011657
  • KONDRAT'EVA G.Y. ET AL.: 'Noncyclic dimer of 4-methyl-2-(dimethylamino)oxazole' IZVESTIYA AKADEMII NAUK SSSR, SERIYA KHIMICHESKAYA no. 7, 1977, pages 1680 - 1682, XP003011658
  • DATABASE CAPLUS [Online] HUENIG S. ET AL.: 'Azo dyes by oxidative coupling. XVIII. Synthesis of 3-substituted 2-thiazolone hydrazones and 2-thiazolone benzenesulfonylhydrazones', XP003011659 Retrieved from STN Database accession no. (1962:46595) & ANN. vol. 647, 1961, pages 66 - 76
   
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