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<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIRO..CY..TRBGCZEEHUPLSK....IS..............................</B001EP><B005EP>J</B005EP><B007EP>DIM360 Ver 2.41 (21 Oct 2013) -  2999001/0</B007EP></eptags></B000><B100><B110>1942105</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20140813</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>06822035.9</B210><B220><date>20061023</date></B220><B240><B241><date>20080508</date></B241><B242><date>20120626</date></B242></B240><B250>ja</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>2005309642</B310><B320><date>20051025</date></B320><B330><ctry>JP</ctry></B330><B310>2006076636</B310><B320><date>20060320</date></B320><B330><ctry>JP</ctry></B330></B300><B400><B405><date>20140813</date><bnum>201433</bnum></B405><B430><date>20080709</date><bnum>200828</bnum></B430><B450><date>20140416</date><bnum>201416</bnum></B450><B452EP><date>20140212</date></B452EP><B480><date>20140813</date><bnum>201433</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 239/14        20060101AFI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/426       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/505       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/506       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/535       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61K  31/54        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61K  31/541       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>A61K  31/5415      20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>A61K  31/55        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>A61K  31/551       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="11"><text>A61K  31/554       20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="12"><text>A61P  25/28        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="13"><text>A61P  43/00        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="14"><text>C07D 239/24        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="15"><text>C07D 265/08        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="16"><text>C07D 277/18        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="17"><text>C07D 279/06        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="18"><text>C07D 279/08        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="19"><text>C07D 281/02        20060101ALI20080530BHEP        </text></classification-ipcr><classification-ipcr sequence="20"><text>C07D 405/04        20060101ALI20080530BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>AMINODIHYDROTHIAZIN-DERIVAT</B542><B541>en</B541><B542>AMINODIHYDROTHIAZINE DERIVATIVE</B542><B541>fr</B541><B542>DERIVE AMINODIHYDROTHIAZINE</B542></B540><B560><B561><text>EP-A1- 0 713 704</text></B561><B561><text>WO-A1-02/096897</text></B561><B561><text>WO-A1-2004/014843</text></B561><B561><text>WO-A1-2004/043916</text></B561><B561><text>WO-A2-2005/111031</text></B561><B561><text>CH-A- 484 184</text></B561><B561><text>JP-A- 08 231 521</text></B561><B561><text>JP-A- 2004 149 429</text></B561><B561><text>JP-A- 2005 509 651</text></B561><B561><text>JP-A- 2005 517 634</text></B561><B561><text>JP-A- 2005 526 005</text></B561><B561><text>JP-A- 2005 531 520</text></B561><B561><text>US-A1- 2005 165 080</text></B561><B562><text>SCHUBERT ET AL.: "Neue Synthesen von 2-Amino-5,6-dihydro-4H-1,3-thiazinen", ARCHIV DER PHARMAZIE, vol. 301, no. 10, 1968, pages 750-762, XP002632395,</text></B562><B562><text>LIEBSCHER J. ET AL.: '2-ARYLIMINO-3-THIAZOLINES - FORMATION OF UNUSUAL TAUTOMERS OF 2-ARYLAMINO-THIAZOLINES - A REVISION' TETRAHEDRON LETTERS vol. 26, no. 35, 1985, pages 4179 - 4180, XP003011652</text></B562><B562><text>GARCIA FERNANDEZ J.M. ET AL.: 'Syntheses and Spectral Properties of beta-Idoureas and 2-Amino-4,4-diphenyl-2-oxazolines' JOURNAL OF HETEROCYCLIC CHEMISTRY vol. 28, no. 3, 1991, pages 777 - 780, XP003011653</text></B562><B562><text>SCHAUMANN. ET AL.: 'Stickstoffhaltige Funfring-Heterocyclen aus Carbodiimiden oder Ketenimine mit 3-Dimethylamino-2H-azirinen' LIEBIGS ANNALEN DER CHEMIE no. 2, 1981, pages 290 - 305, XP003011654</text></B562><B562><text>GARCIA FERNANDEZ J.M. ET AL.: 'Syntheses of beta-iodourea derivatives of carbohydrates and glycosylamino-oxazolines' CARBOHYDRATE RESEARCH vol. 216, 1991, pages 21 - 32, XP003011655</text></B562><B562><text>COHEN N. ET AL.: 'Synthesis of 2-Amino-5-, 6-dihydro-4H-1,3-thiazines and Related Compounds by Acid Catalyzed Cyclization of Allylic Isothiuronium Salts' JOURNAL OF HETEROCYCLIC CHEMISTRY vol. 14, no. 5, 1977, pages 717 - 723, XP003011656</text></B562><B562><text>CAMBIE R.C. ET AL.: 'vic-Iodothiocyanates and Iodoisothiocyanates. Part 2. New Syntheses of Thiazolidin-2-ones and 2-Amino-2-thiazolines' JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS I no. 3, 1979, pages 765 - 770, XP003011657</text></B562><B562><text>KONDRAT'EVA G.Y. ET AL.: 'Noncyclic dimer of 4-methyl-2-(dimethylamino)oxazole' IZVESTIYA AKADEMII NAUK SSSR, SERIYA KHIMICHESKAYA no. 7, 1977, pages 1680 - 1682, XP003011658</text></B562><B562><text>DATABASE CAPLUS [Online] HUENIG S. ET AL.: 'Azo dyes by oxidative coupling. XVIII. Synthesis of 3-substituted 2-thiazolone hydrazones and 2-thiazolone benzenesulfonylhydrazones', XP003011659 Retrieved from STN Database accession no. (1962:46595) &amp; ANN. vol. 647, 1961, pages 66 - 76</text></B562><B565EP><date>20110516</date></B565EP></B560></B500><B600><B620EP><parent><cdoc><dnum><anum>13150548.9</anum><pnum>2612854</pnum></dnum><date>20130108</date></cdoc><cdoc><dnum><anum>13150550.5</anum><pnum>2597087</pnum></dnum><date>20130108</date></cdoc></parent></B620EP></B600><B700><B720><B721><snm>KOBAYASHI, Naotake</snm><adr><str>c/o Shionogi &amp; Co., Ltd. 12-4, Sagisu 5-chome, Fuk
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