(19)
(11) EP 1 963 284 A1

(12)

(43) Date of publication:
03.09.2008 Bulletin 2008/36

(21) Application number: 06830421.1

(22) Date of filing: 06.12.2006
(51) International Patent Classification (IPC): 
C07D 239/95(2006.01)
C07D 401/04(2006.01)
(86) International application number:
PCT/EP2006/069380
(87) International publication number:
WO 2007/065913 (14.06.2007 Gazette 2007/24)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

(30) Priority: 07.12.2005 DK 200501732
08.12.2005 US 748221 P

(71) Applicant: NeuroSearch A/S
2750 Ballerup (DK)

(72) Inventors:
  • SØRENSEN, Ulrik, Svane
    DK-2750 Ballerup (DK)
  • ERIKSEN, Birgitte, L.
    DK-2750 Ballerup (DK)
  • TEUBER, Lene
    DK-3500 Værløse (DK)
  • PETERS, Dan
    DK-2750 Ballerup (DK)
  • STRØBÆK, Dorte
    DK-2750 Ballerup (DK)
  • JOHANSEN, Tina, Holm
    DK-2765 Smorum (DK)
  • CHRISTOPHERSEN, Palle
    DK-2750 Ballerup (DK)

(74) Representative: Madsen, Inger Margrethe Schelde et al
NeuroSearch A/S Patent Department 93 Pederstrupvej
2750 Ballerup
2750 Ballerup (DK)

   


(54) NOVEL QUINAZOLINE-2,4-DIAMINE DERIVATIVES AND THEIR USE AS MODULATORS OF SMALL-CONDUCTANCE CALCIUM-ACTIVATED POTASSIUM CHANNELS