3-PYRIDINYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO - Patent 2004627

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(11)

EP 2 004 627 A2

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(88)	Date of publication A3:
	03.01.2008

(43)	Date of publication:
	24.12.2008 Bulletin 2008/52

(21)	Application number: 07774984.4

(22)	Date of filing: 09.04.2007

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International Patent Classification (IPC):

C07D 401/04^(2006.01)
C07D 413/14^(2006.01)
A61P 9/00^(2006.01)

C07D 401/14^(2006.01)
A61K 31/4439^(2006.01)

(86)	International application number:
	PCT/US2007/008718

(87)	International publication number:
	WO 2007/120600 (25.10.2007 Gazette 2007/43)

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR
	Designated Extension States:
	AL BA HR MK RS

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Priority:

10.04.2006 US 790686 P

(71)	Applicant: Arena Pharmaceuticals, Inc.
	San Diego, CA 92121-3223 (US)

(72)	Inventors:
	DOSA, Peter I. San Diego, CA 92126 (US) TEEGARDEN, Bradley San Diego, CA 92131 (US)

(74)	Representative: Wytenburg, Wilhelmus Johannes et al
	Mewburn Ellis LLP York House 23 Kingsway London WC2B 6HP London WC2B 6HP (GB)

(54)	3-PYRIDINYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO