(19)
(11) EP 2 054 391 A1

(12)

(43) Date of publication:
06.05.2009 Bulletin 2009/19

(21) Application number: 06780412.0

(22) Date of filing: 17.08.2006
(51) International Patent Classification (IPC): 
C07D 239/47(2006.01)
(86) International application number:
PCT/IL2006/000958
(87) International publication number:
WO 2008/020425 (21.02.2008 Gazette 2008/08)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
Designated Extension States:
AL BA HR MK RS

(71) Applicant: CHEMAGIS LTD.
51200 Bnei-Brak (IL)

(72) Inventors:
  • ADIN, Itai
    84684 Beer-sheva (IL)
  • IUSTAIN, Carmen
    84750 Beer-sheva (IL)
  • WEISMAN, Alexander
    70500 Kiryat-ekron (IL)
  • ARAD, Oded
    76303 Rechovot (IL)
  • KASPI, Joseph
    53201 Givatayim (IL)

(74) Representative: Albrecht, Thomas 
Kraus & Weisert Patent- und Rechtsanwälte Thomas-Wimmer-Ring 15
80539 München
80539 München (DE)

   


(54) CRYSTALLINE MOXONIDINE COMPRISING SINGLE TAUTOMER AND PREPARATION PROCESS THEREFOR