TRIAZOLE DERIVATIVES AS KINASE INHIBITORS

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EP 2 057 158 B8

(12)	CORRECTED EUROPEAN PATENT SPECIFICATION
	Note: Bibliography reflects the latest situation

(15)	Correction information:
	Corrected version no 1 (W1 B1)

(48)	Corrigendum issued on:
	30.09.2015 Bulletin 2015/40

(45)	Mention of the grant of the patent:
	12.08.2015 Bulletin 2015/33

(21)	Application number: 07803060.8

(22)	Date of filing: 30.08.2007

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International Patent Classification (IPC):

C07D 471/04^(2006.01)
A61P 29/00^(2006.01)
A61P 35/00^(2006.01)

A61K 31/437^(2006.01)
A61P 37/00^(2006.01)

(86)	International application number:
	PCT/EP2007/059051

(87)	International publication number:
	WO 2008/025821 (06.03.2008 Gazette 2008/10)

(54)	TRIAZOLE DERIVATIVES AS KINASE INHIBITORS TRIAZOLDERIVATE ALS KINASEINHIBITOREN DÉRIVÉS DE TRIAZOLE EN TANT QU'INHIBITEURS DE KINASE

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR

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Priority:

30.08.2006 EP 06119831
23.05.2007 EP 07108769

(43)	Date of publication of application:
	13.05.2009 Bulletin 2009/20

(73)	Proprietor: Cellzome Limited
	Brentford, Middlesex TW8 9GS (GB)

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Inventors:

WILSON, Francis
Herts Hertfordshire AL 7 AQJ (GB)
RAMSDEN, Nigel
Royston, Herts Hertfordshire SG8 7QP (GB)
BELL, Kathryn
London London EC1R 5HP (GB)
CANSFIELD, Andrew
Harston Cambridgeshire CB22 7QT (GB)
BURCKHARDT, Svenja
Newmarket CB8 9QG (GB)
TAYLOR, Jess
Stotfold, Hitchin Hertfordshire SG5 4PJ (GB)
SUNOSE, Mihiro
Pampisford Cambridgeshire CB22 3EW (GB)
MIDDLEMISS, David
Bishops Stortford Hertfordshire CM23 33NF (GB)

(74)	Representative: Shore, Andrew David
	GlaxoSmithKline Global Patents (CN925.1) 980 Great West Road Brentford, Middlesex TW8 9GS Brentford, Middlesex TW8 9GS (GB)

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References cited: :

WO-A-03/010167
WO-A1-96/31517
WO-A2-2006/018735

WO-A-2004/072072
WO-A1-2007/095588
WO-A2-2006/038116

NETTEKOVEN, MATTHIAS ET AL: "Synthetic access to 2-amido-5-aryl-8-methoxy-triazolopyridine and 2-amido-5-morpholino-8-methoxy-triazolopyr idine derivatives as potential inhibitors of the adenosine receptor subtypes" SYNTHESIS , (11), 1649-1652 CODEN: SYNTBF; ISSN: 0039-7881, 2003, XP002416826
YAMAZAKI, CHIJI ET AL: "Cyclization of isothiosemicarbazones. Part 10. A novel route to 2-amino[1,2,4]triazolo[1,5-a]pyridine derivatives" JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 1: ORGANIC AND BIO-ORGANIC CHEMISTRY (1972-1999) , (7), 825-8 CODEN: JCPRB4; ISSN: 0300-922X, 1994, XP002416827


	Remarks:
	The file contains technical information submitted after the application was filed and not included in this specification

Note: Within nine months from the publication of the mention of the grant of the European patent, any person may give notice to the European Patent Office of opposition to the European patent granted. Notice of opposition shall be filed in a written reasoned statement. It shall not be deemed to have been filed until the opposition fee has been paid. (Art. 99(1) European Patent Convention).