(19)
(11) EP 2 099 814 A1

(12)

(43) Date of publication:
16.09.2009 Bulletin 2009/38

(21) Application number: 07847383.2

(22) Date of filing: 27.11.2007
(51) International Patent Classification (IPC): 
C07J 41/00(2006.01)
C07J 51/00(2006.01)
A61K 31/58(2006.01)
A61P 5/32(2006.01)
C07J 43/00(2006.01)
A61K 31/565(2006.01)
A61K 31/566(2006.01)
(86) International application number:
PCT/EP2007/062856
(87) International publication number:
WO 2008/065100 (05.06.2008 Gazette 2008/23)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR

(30) Priority: 30.11.2006 EP 06125138

(71) Applicant: Solvay Pharmaceuticals GmbH
30173 Hannover (DE)

(72) Inventors:
  • MESSINGER, Josef
    30173 Hannover (DE)
  • HUSEN, Bettina
    30173 Hannover (DE)
  • SCHOEN, Uwe
    30173 Hannover (DE)
  • THOLE, Heinrich-Hubert
    30173 Hannover (DE)
  • KOSKIMIES, Pasi
    30173 Hannover (DE)
  • UNKILA, Mikko
    30173 Hannover (DE)

(74) Representative: Gosmann, Martin et al
Solvay Pharmaceuticals GmbH Hans-Böckler-Allee 20
30173 Hannover
30173 Hannover (DE)

   


(54) SUBSTITUTED ESTRATRIEN DERIVATIVES AS 17BETA HSD INHIBITORS