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<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIRO..CY..TRBGCZEEHUPLSK..HRIS..MTNO........................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>JDIM360 Ver 1.28 (29 Oct 2014) -  2999001/0</B007EP></eptags></B000><B100><B110>2137191</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20160608</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>08742363.8</B210><B220><date>20080328</date></B220><B240><B241><date>20091013</date></B241><B242><date>20140917</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>921123 P</B310><B320><date>20070329</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20160608</date><bnum>201623</bnum></B405><B430><date>20091230</date><bnum>200953</bnum></B430><B450><date>20160302</date><bnum>201609</bnum></B450><B452EP><date>20150821</date></B452EP><B480><date>20160608</date><bnum>201623</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 489/04        20060101AFI20081021BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/439       20060101ALI20081021BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61P  43/00        20060101ALI20081021BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>ANTAGONISTEN DER PERIPHEREN OPIOIDREZEPTOREN UND IHRE VERWENDUNG</B542><B541>en</B541><B542>PERIPHERAL OPIOID RECEPTOR ANTAGONISTS AND USES THEREOF</B542><B541>fr</B541><B542>ANTAGONISTES DE RÉCEPTEURS OPIOÏDES PÉRIPHÉRIQUES, ET LEURS UTILISATIONS</B542></B540><B560><B561><text>WO-A-2006/127899</text></B561><B562><text>UWAI, KOJI ET AL.: BIOORGANIC &amp; MEDICINAL CHEMISTRY, vol. 12, 2004, pages 417-421, XP002499242</text></B562><B562><text>LAZAR S ET AL: "SYNTHESIS AND BIOLOGICAL ACTIVITY OF THE PHOSPHATE AND SULFATE ESTERS OF NALOXONE AND NALTREXONE" EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, EDITIONS SCIENTIFIQUE ELSEVIER, PARIS, FR, vol. 29, no. 1, 1 January 1994 (1994-01-01), pages 45-54, XP009084006 ISSN: 0223-5234</text></B562><B562><text>MALSPEIS L ET AL: "METABOLIC REDUCTION OF NALTEXONE I. SYNTHESIS, SEPARATION AND CHARACTERIZATION OF NALOXONE AND NALTREXONE REDUCTION PRODUCTS AND QUALITATIVE ASSAY OF URINE AND BILE FOLLOWING ADMINISTRATION OF NALTREXONE, ALPHA-NALTREXOL, OR BETA-NALTREXOL" RESEARCH COMMUNICATIONS IN CHEMICAL PATHOLOGY AND PHARMACOLOGY, PJD PUBLICATIONS LTD., WESTBURY, NY, US, vol. 12, no. 1, 1 September 1975 (1975-09-01), pages 43-65, XP008097305 ISSN: 0034-5164</text></B562></B560></B500><B600><B620EP><parent><cdoc><dnum><anum>16155008.2</anum></dnum><date>20160210</date></cdoc></parent></B620EP></B600><B700><B720><B721><snm>AVEY, Alfred, A.</snm><adr><str>2568 Tarris View Drive</str><city>Eugene, OR 07405</city><ctry>US</ctry></adr></B721><B721><snm>PEREZ, Julio</snm><adr><str>273D, South Broadway</str><city>Tarrytown, NY 10591</city><ctry>US</ctry></adr></B721><B721><snm>DOSHAN, Harold, D.</snm><adr><str>18 Griffith Road</str><city>Riverside, CT 06878</city><ctry>US</ctry></adr></B721><B721><snm>CHANDRASEKARAN, Appavu</snm><adr><str>35 Thoreau Drive</str><city>Plainsboro, NJ 08536</city><ctry>US</ctry></adr></B721><B721><snm>ROTSHTEYN, Yakov</snm><adr><str>5 Kasch Court</str><city>Monroe, NY 10950</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>Progenics Pharmaceuticals, Inc.</snm><iid>101016906</iid><irf>TXR/60250EP1</irf><adr><str>777 Old Saw Mill River Road</str><city>Tarrytown, NY 10591</city><ctry>US</ctry></adr></B731><B731><snm>Wyeth LLC (Formerly Known As Wyeth)</snm><iid>101578087</iid><irf>TXR/60250EP1</irf><adr><str>235 East 42nd Street</str><city>New York, NY 10017</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Russell, Tim</snm><iid>101291355</iid><adr><str>Venner Shipley LLP 
200 Aldersgate</str><city>London EC1A 4HD</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>US2008004109</anum></dnum><date>20080328</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2008121348</pnum></dnum><date>20081009</date><bnum>200841</bnum></B871></B870></B800></SDOBI>
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