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EP 2 152 708 A1

(12)

(43) Date of publication: 17.02.2010 Bulletin 2010/07 (21) Application number: 07797679.3 (22) Date of filing: 23.05.2007

(51) International Patent Classification (IPC):  C07D 471/04(2006.01) C07D 487/04(2006.01) A61P 37/06(2006.01) C07D 473/00(2006.01) A61K 31/522(2006.01) (86) International application number: PCT/US2007/069530 (87) International publication number: WO 2008/143674 (27.11.2008 Gazette 2008/48)

(84) Designated Contracting States: AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR Designated Extension States: AL BA HR MK RS (71) Applicant: Pharmacopeia, LLC Princetown NJ 08543 (US)	(72) Inventors: ROUGHTEN, Andrew Plainsboro, NJ 08536 (US) RONG, Yajing Monmouth Junction, NJ 08852 (US) HO, Koc Kan West Windsor, NJ 08550 (US) OHLMEYER, Michael Plainsboro, NJ 08536 (US) DILLER, David East Windsor, NJ 08520 (US) (74) Representative: Jaap, David Robert et al P.O. Box 20 5340 BH Oss 5340 BH Oss (NL)