(19)
(11) EP 2 187 893 A2

(12)

(88) Date of publication A3:
01.04.2010

(43) Date of publication:
26.05.2010 Bulletin 2010/21

(21) Application number: 09700012.9

(22) Date of filing: 05.03.2009
(51) International Patent Classification (IPC): 
A61K 31/69(2006.01)
(86) International application number:
PCT/US2009/036250
(87) International publication number:
WO 2009/111676 (11.09.2009 Gazette 2009/37)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA RS

(30) Priority: 06.03.2008 US 34371 P
12.05.2008 US 52637 P
04.09.2008 US 94406 P
16.10.2008 US 105990 P

(71) Applicant: Anacor Pharmaceuticals, Inc.
Palo Alto, CA 94303 (US)

(72) Inventors:
  • AKAMA, Tsutomu
    Sunnyvale, CA 94087 (US)
  • ZHANG, Yong-kang
    San Jose, CA 95130 (US)
  • DING, Charles Z.
    Palo Alto, CA 94303 (US)
  • PLATTNER, Jacob J.
    Berkeley, CA 94705 (US)
  • MAPLES, Kirk R.
    San Jose, CA 95132 (US)
  • FREUND, Yvonne
    Los Alto, CA 94024 (US)
  • SANDERS, Virginia
    San Francisco, CA 94110 (US)
  • XIA, Yi
    Palo Alto, CA 94306 (US)
  • BAKER, Stephen J.
    Mountain View, CA 94040 (US)
  • NIEMANN, James A.
    Sherwood Park Alberta, T8H 2P8 (CA)
  • Lu, Xiaosong
    Edmonton Alberta, T6R 0J9 (CA)
  • SALES, Marcelo
    Edmonton Alberta, T6E 2T3 (CA)
  • SHARMA, Rashmi
    Edmonton Alberta, T6T 0A7 (CA)
  • SINGH, Rajeshwar
    Edmonton Alberta, T6R 2Y1 (CA)
  • JACOBS, Robert
    Durham, NC 27713 (US)
  • CHEN, Daitao
    Durham, NC 27713 (US)
  • ALLEY, Michael Richard Kevin
    Santa Clara, CA 95051 (US)

(74) Representative: Harrison Goddard Foote 
Belgrave Hall Belgrave Street
Leeds LS2 8DD
Leeds LS2 8DD (GB)

   


(54) BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS