(19)
(11) EP 2 194 975 A2

(12)

(88) Date of publication A3:
26.03.2009

(43) Date of publication:
16.06.2010 Bulletin 2010/24

(21) Application number: 08826259.7

(22) Date of filing: 11.07.2008
(51) International Patent Classification (IPC): 
A61K 31/15(2006.01)
A61P 9/10(2006.01)
A61P 25/28(2006.01)
(86) International application number:
PCT/US2008/069878
(87) International publication number:
WO 2009/009768 (15.01.2009 Gazette 2009/03)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA MK RS

(30) Priority: 12.07.2007 US 777264
12.07.2007 US 777266
19.07.2007 US 950724 P
19.07.2007 US 950810 P

(71) Applicant: Acumen Pharmaceuticals, Inc.
Livermore, CA 94551 (US)

(72) Inventors:
  • LOOK, Gary Charles
    Santa Clara, California 95051 (US)
  • SCHULTZ, Lauri
    Batavia, Illinois 60510 (US)
  • POLOZOV, Alexandre Mikhaylovich
    Naperville, Illinois 60565 (US)
  • BHAGAT, Nikhil
    Aurora, Illinois 60503-5762 (US)
  • WANG, Jian
    San Diego, California 92129 (US)
  • ZEMBOWER, David E.
    La Grange, Illinois 60525 (US)
  • GOURE, William, F.
    Livermore, California 94551 (US)
  • PRAY, Todd
    San Mateo, California 94554 (US)
  • KRAFFT, Grant, A.
    Glenview, Illinois 60025 (US)

(74) Representative: Wibbelmann, Jobst 
Wuesthoff & Wuesthoff Patent- und Rechtsanwälte Schweigerstrasse 2
81541 München
81541 München (DE)

   


(54) METHODS OF INHIBITING THE FORMATION OF AMYLOID-ß DIFFUSABLE LIGANDS USING A ACYLHYDRAZIDE COMPOUNDS