<?xml version="1.0" encoding="UTF-8"?>
<!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.5//EN" "ep-patent-document-v1-5.dtd">
<ep-patent-document id="EP08846682B8W1" file="EP08846682W1B8.xml" lang="en" country="EP" doc-number="2209377" kind="B8" correction-code="W1" date-publ="20180905" status="c" dtd-version="ep-patent-document-v1-5">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIRO..CY..TRBGCZEEHUPLSK..HRIS..MTNO........................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 0.1.63 (23 May 2017) -  2999001/0</B007EP></eptags></B000><B100><B110>2209377</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20180905</date></B140><B150><B151>W1</B151><B153>72 73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>08846682.6</B210><B220><date>20081106</date></B220><B240><B241><date>20100603</date></B241><B242><date>20130418</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>985972 P</B310><B320><date>20071106</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20180905</date><bnum>201836</bnum></B405><B430><date>20100728</date><bnum>201030</bnum></B430><B450><date>20180502</date><bnum>201818</bnum></B450><B452EP><date>20171208</date></B452EP><B480><date>20180905</date><bnum>201836</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>A01N  45/00        20060101AFI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/00        20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/592       20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/593       20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>C12Q   1/02        20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61P   1/16        20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61P   1/18        20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>G01N  33/82        20060101ALI20171113BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>G01N  33/50        20060101ALI20171113BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>VERWENDUNG VON VITAMINREZEPTORAGONISTEN UND VORSTUFEN FÜR DIE BEHANDLUNG VON FIBROSE</B542><B541>en</B541><B542>USE OF VITAMIN D RECEPTOR AGONISTS AND PRECURSORS TO TREAT FIBROSIS</B542><B541>fr</B541><B542>UTILISATION D'AGONISTES ET DE PRÉCURSEURS DE RÉCEPTEURS DE LA VITAMINE D POUR TRAITER LA FIBROSE</B542></B540><B560><B561><text>EP-A1- 0 682 879</text></B561><B561><text>US-A1- 2005 009 793</text></B561><B561><text>US-A1- 2005 124 591</text></B561><B561><text>US-A1- 2006 074 109</text></B561><B561><text>US-A1- 2006 135 610</text></B561><B561><text>US-A1- 2006 240 150</text></B561><B562><text>TAN ET AL: "Therapeutic role and potential mechanisms of active Vitamin D in renal interstitial fibrosis" JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, ELSEVIER SCIENCE LTD., OXFORD, GB LNKD- DOI:10.1016/J.JSBMB.2006.11.011, vol. 103, no. 3-5, 15 March 2007 (2007-03-15), pages 491-496, XP022275094 ISSN: 0960-0760</text></B562><B562><text>TAN XIAOYUE ET AL: "Paricalcitol attenuates renal interstitial fibrosis in obstructive nephropathy" JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY, vol. 17, no. 12, December 2006 (2006-12), pages 3382-3393, XP002605885 ISSN: 1046-6673</text></B562><B562><text>GASCON-BARRE ET AL.: 'The normal liver harbors the vitamin D nuclear receptor in nonparenchymal and biliary epithelial cells.' HEPATOLOGY vol. 37, no. 5, 2003, pages 1034 - 1042</text></B562><B562><text>OMARY ET AL.: 'The pancreatic stellate cell: a star on the rise in pancreatic diseases.' JOURNAL OF CLINICAL INVESTIGATION vol. 117, no. 1, January 2007, pages 50 - 59</text></B562><B562><text>ZEHNDER ET AL.: 'Expression of 25-hydroxyvitamin D3-lalpha-hydroxylase in the human kidney.' J AM SOC NEPHROL vol. 10, 1999, pages 2465 - 2473</text></B562><B562><text>JOHNSON ET AL.: 'The activated mesangial cell: a glomerulat myofibroblast?' JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY vol. 2, no. SUP 02, 1992, pages S190 - S197</text></B562><B562><text>CAO ET AL.: 'Leptin stimulates tissue inhibitor of metalloproteinase-1 in human hepatic stellate cells.' JOURNAL OF BIOLOGICAL CHEMISTRY vol. 279, no. 6, 2004, pages 4292 - 4304</text></B562><B562><text>J A MCCARROLL: "Vitamin A inhibits pancreatic stellate cell activation: implications for treatment of pancreatic fibrosis", GUT, vol. 55, no. 1, 1 January 2006 (2006-01-01), pages 79-89, XP055395056, UK ISSN: 0017-5749, DOI: 10.1136/gut.2005.064543</text></B562><B565EP><date>20101109</date></B565EP></B560></B500><B700><B720><B721><snm>EVANS, Ronald, M.</snm><adr><str>1471 CottontailLane</str><city>La Jolla
CA 92037</city><ctry>US</ctry></adr></B721><B721><snm>DOWNES, Michael</snm><adr><str>2730 Havasupai Avenue</str><city>San Diego
CA 92117</city><ctry>US</ctry></adr></B721><B721><snm>LIDDLE, Christopher</snm><adr><str>4 Rebecca Place</str><city>Tura Beach
New South Wales 2548</city><ctry>AU</ctry></adr></B721></B720><B730><B731><snm>The Salk Institute For Biological Studies</snm><iid>101113640</iid><irf>3818P/EP</irf><adr><str>10010 N. Torrey Pines Road</str><city>La Jolla, CA 92037-1099</city><ctry>US</ctry></adr></B731><B731><snm>University of Sydney</snm><iid>101754334</iid><irf>3818P/EP</irf><adr><city>NSW 2000</city><ctry>AU</ctry></adr></B731></B730><B740><B741><snm>Harrison IP Limited</snm><iid>101296927</iid><adr><str>3 Ebor House 
Millfield Lane</str><city>Nether Poppleton, York YO26 6QY</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>US2008082691</anum></dnum><date>20081106</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2009061961</pnum></dnum><date>20090514</date><bnum>200920</bnum></B871></B870></B800></SDOBI>
</ep-patent-document>
