BICYCLIC HETEROCYCLE DERIVATIVES AND THEIR USE AS MODULATORS OF THE ACTIVITY OF GPR119

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EP 2 217 596 B8

(12)	CORRECTED EUROPEAN PATENT SPECIFICATION
	Note: Bibliography reflects the latest situation

(15)	Correction information:
	Corrected version no 1 (W1 B1)

(48)	Corrigendum issued on:
	20.11.2013 Bulletin 2013/47

(45)	Mention of the grant of the patent:
	30.01.2013 Bulletin 2013/05

(21)	Application number: 08832779.6

(22)	Date of filing: 20.10.2008

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International Patent Classification (IPC):

C07D 451/06^(2006.01)
C07D 498/08^(2006.01)
C07D 491/08^(2006.01)
A61K 31/439^(2006.01)
A61K 31/537^(2006.01)
C07D 401/14^(2006.01)

C07D 471/08^(2006.01)
C07D 487/08^(2006.01)
A61K 31/46^(2006.01)
A61K 31/506^(2006.01)
A61P 3/00^(2006.01)
C07D 495/08^(2006.01)

(86)	International application number:
	PCT/US2008/080462

(87)	International publication number:
	WO 2009/055331 (30.04.2009 Gazette 2009/18)

(54)	BICYCLIC HETEROCYCLE DERIVATIVES AND THEIR USE AS MODULATORS OF THE ACTIVITY OF GPR119 BICYCLISCHE HETEROCYCLISCHE DERIVATE UND IHRE VERWENDUNG ALS MODULATOREN DER AKTIVITÄT VON GPR 119 DÉRIVÉS HÉTÉROCYCLIQUES BICYCLIQUES ET LEUR UTILISATION EN TANT QUE MODULATEURS DE L'ACTIVITE DU GPR 119

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
	Designated Extension States:
	AL BA MK RS

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Priority:

22.10.2007 US 981677 P

(43)	Date of publication of application:
	18.08.2010 Bulletin 2010/33

(73)	Proprietor: Merck Sharp & Dohme Corp.
	Rahway, NJ 07065-0907 (US)

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Inventors:

XIA, Yan
Edison New Jersey 08820 (US)
BOYLE, Craig, D.
Branchburg New Jersey 08876 (US)
GREENLEE, William, J.
Teaneck New Jersey 07666 (US)
CHACKALAMANNIL, Samuel
Califon New Jersey 07830 (US)
JAYNE, Charles, Lee
Staten Island New York 10305 (US)
STAMFORD, Andrew, W.
Chatham Township New Jersey 07928 (US)
DAI, Xing
Scotch Plains New Jersey 07076 (US)
HARRIS, Joel, M.
Summit New Jersey 07901 (US)
NEUSTADT, Bernard, R.
West Orange New Jersey 07052 (US)
NEELAMKAVIL, Santhosh, Francis
Scotch Plains New Jersey 07076 (US)
SHAH, Unmesh, G.
Greenbrook New Jersey 08812 (US)
LANKIN, Claire, M.
High Bridge New Jersey 08829 (US)
LIU, Hong
Hillsborough New Jersey 08844 (US)

(74)	Representative: Jaap, David Robert et al
	Merck & Co., Inc. Hertford Road Hoddesdon, Herts EN11 9BU Hoddesdon, Herts EN11 9BU (GB)

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References cited: :

WO-A-2005/007647

Note: Within nine months from the publication of the mention of the grant of the European patent, any person may give notice to the European Patent Office of opposition to the European patent granted. Notice of opposition shall be filed in a written reasoned statement. It shall not be deemed to have been filed until the opposition fee has been paid. (Art. 99(1) European Patent Convention).