(19)
(11) EP 2 231 646 A1

(12)

(43) Date of publication:
29.09.2010 Bulletin 2010/39

(21) Application number: 08859397.5

(22) Date of filing: 10.12.2008
(51) International Patent Classification (IPC): 
C07D 401/14(2006.01)
A61P 5/04(2006.01)
 A61K 31/33(2006.01)
(86) International application number:
PCT/US2008/086131
(87) International publication number:
WO 2009/076387 (18.06.2009 Gazette 2009/25)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA MK RS

(30) Priority: 10.12.2007 US 12525

(71) Applicant: GlaxoSmithKline LLC
Philadelphia, PA 19102 (US)

(72) Inventors:
  • ALLEN, Scott
    Research Triangle Park, North Carolina 27709 (US)
  • BLACKWELL III, William C.
    Research Triangle Park, North Carolina 27709 (US)
  • BOROS, Eric
    Research Triangle Park, North Carolina 27709 (US)
  • COLLINS, Jon L
    Research Triangle Park, North Carolina 27709 (US)
  • HERTZOG, Don
    Research Triangle Park, NorthCarolina 27709 (US)
  • LIANG, Xi
    Research Triangle Park, North Carolina 27709 (US)
  • RAY, John
    Research Triangle Park, North Carolina 27709 (US)
  • REISTER, Steven Michael
    Research Triangle Park, North Carolina 27709 (US)
  • SAMANO, Vicente
    Research Triangle Park, North Carolina 27709 (US)
  • SHERRILL, Ron
    Research Triangle Park, North Carolina 27709 (US)

(74) Representative: Goddard, Carolyn Janice et al
GlaxoSmithKline Corporate Intellectual Property (CN925.1) 980 Great West Road Brentford
Middlesex TW8 9GS
Middlesex TW8 9GS (GB)

   


(54) BIS-PYRIDYLPYRIDONES AS MELANIN-CONCENTRATING HORMONE RECEPTOR 1 ANTAGONISTS