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EP 2 235 036 A1

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(43) Date of publication: 06.10.2010 Bulletin 2010/40 (21) Application number: 09706942.1 (22) Date of filing: 28.01.2009

(51) International Patent Classification (IPC):  C07J 63/00(2006.01) A61P 35/00(2006.01) A61K 31/70(2006.01) (86) International application number: PCT/CZ2009/000007 (87) International publication number: WO 2009/094958 (06.08.2009 Gazette 2009/32)

(84) Designated Contracting States: AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR Designated Extension States: AL BA RS (30) Priority: 30.01.2008 CZ 20080051 (71) Applicants: Universita Palackeho v Olomouci 771 47 Olomouc (CZ) Institute Of Organic Chemistry, Polish Academy Of Sciences 01-224 Warszawa (PL) Bio Apex S.r.o. 779 00 Olomouc (CZ)

(72) Inventors: PAKULSKI, Zbigniew Andrzej PL-02-796 Warszawa (PL) CMOCH, Piotr PL-01-057 Warszawa (PL) OKLESTKOVA, Jana 798 14 Olsany u Prostejova (CZ) STRNAD, Miroslav 779 00 Olomouc (CZ) (74) Representative: Gabrielova, Marta  Inventia s.r.o. Na Belidle 3 150 00 Praha 5 150 00 Praha 5 (CZ)