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<ep-patent-document id="EP09713314B8W1" file="EP09713314W1B8.xml" lang="en" country="EP" doc-number="2254880" kind="B8" correction-code="W1" date-publ="20160921" status="c" dtd-version="ep-patent-document-v1-5">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCY..TRBGCZEEHUPLSK..HRIS..MTNO........................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>JDIM360 Ver 1.28 (29 Oct 2014) -  2999001/0</B007EP></eptags></B000><B100><B110>2254880</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20160921</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>09713314.4</B210><B220><date>20090223</date></B220><B240><B241><date>20100921</date></B241><B242><date>20121123</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>30446 P</B310><B320><date>20080221</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20160921</date><bnum>201638</bnum></B405><B430><date>20101201</date><bnum>201048</bnum></B430><B450><date>20160817</date><bnum>201633</bnum></B450><B452EP><date>20151105</date></B452EP><B480><date>20160921</date><bnum>201638</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 313/00        20060101AFI20120110BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 315/00        20060101ALI20120110BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/365       20060101ALI20120110BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>Als Therapeutika geeignete makrocyclische Prodrugverbindungen</B542><B541>en</B541><B542>Macrocyclic prodrug compounds useful as therapeutics</B542><B541>fr</B541><B542>Composés de promédicaments macrocycliques utilisés comme agents thérapeutiques</B542></B540><B560><B561><text>EP-A1- 0 460 950</text></B561><B561><text>EP-A1- 0 823 429</text></B561><B561><text>WO-A1-2004/024142</text></B561><B561><text>JP-A- 9 202 781</text></B561><B561><text>JP-A- 10 265 381</text></B561><B561><text>JP-A- 2003 113 183</text></B561><B561><text>US-A1- 2005 182 129</text></B561><B562><text>FRANZ BRACHER ET AL.: 'The total synthesis of both enantiomers of the macrocyclic lactone zearalane.' EUR.J.ORG.CHEM. 2001, pages 4701 - 4704, XP008141388</text></B562><B565EP><date>20120116</date></B565EP></B560></B500><B700><B720><B721><snm>HECK, James</snm><adr><str>c/o Nexgenix Pharmaceuticals
152 West 57th Street
Suite 11B</str><city>New York, NY 10019</city><ctry>US</ctry></adr></B721><B721><snm>WINSSINGER, Nicolas</snm><adr><str>30 rue Jean-Jacques Rousseau</str><city>F-67000 Strasbourg</city><ctry>FR</ctry></adr></B721><B721><snm>CHABALA, John C.</snm><adr><str>c/o Nexgenix Pharmaceuticals
152 West 57th Street
Suite 11B</str><city>New York, NY 10019</city><ctry>US</ctry></adr></B721><B721><snm>BARLUENGA, Sofia</snm><adr><str>30 rue Jean-Jacques Rousseau</str><city>F-67000 Strasbourg</city><ctry>FR</ctry></adr></B721><B721><snm>CHEN, Ruihong</snm><adr><str>c/o Nexgenix Pharmaceuticals
152 West 57th Street
Suite 11B</str><city>New York, NY 10019</city><ctry>US</ctry></adr></B721><B721><snm>RUBENSTEIN, Allan</snm><adr><str>c/o Nexgenix Pharmaceuticals
152 West 57th Street
Suite 11B</str><city>New York, NY 10019</city><ctry>US</ctry></adr></B721><B721><snm>YU, Jin-Chen</snm><adr><str>c/o Nexgenix Pharmaceuticals
152 West 57th Street
Suite 11B</str><city>New York, NY 10019</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>OncoSynergy, Inc.</snm><iid>101606526</iid><irf>S2816 EP S3</irf><adr><str>409 Illinois St., Room 3041</str><city>San Francisco, CA 94158</city><ctry>US</ctry></adr></B731><B731><snm>Université de Strasbourg</snm><iid>101133415</iid><irf>S2816 EP S3</irf><adr><str>4, rue Blaise Pascal</str><city>67070 Strasbourg</city><ctry>FR</ctry></adr></B731></B730><B740><B741><snm>Vossius &amp; Partner 
Patentanwälte Rechtsanwälte mbB</snm><iid>100751388</iid><adr><str>Siebertstrasse 3</str><city>81675 München</city><ctry>DE</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MK</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>US2009034878</anum></dnum><date>20090223</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2009105755</pnum></dnum><date>20090827</date><bnum>200935</bnum></B871></B870></B800></SDOBI>
</ep-patent-document>
