(19)
(11) EP 2 262 370 A1

(12)

(43) Date of publication:
22.12.2010 Bulletin 2010/51

(21) Application number: 08744863.5

(22) Date of filing: 01.04.2008
(51) International Patent Classification (IPC): 
A01N 57/00(2006.01)
A61K 31/66(2006.01)
(86) International application number:
PCT/US2008/059025
(87) International publication number:
WO 2009/123623 (08.10.2009 Gazette 2009/41)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA MK RS

(71) Applicant: Virobay, Inc.
Menlo Park, CA 94025 (US)

(72) Inventors:
  • LINK, John, O.
    San Francisco CA 94110 (US)
  • MOSSMAN, Craig, J.
    Saratoga, CA 95070 (US)
  • LIU, Jie
    Shanghai 201203 (CN)
  • WOO, Soon Hyung
    Vista CA 92081-8356 (US)

(74) Representative: Campbell, Patrick John Henry 
J.A. Kemp & Co. 14 South Square Gray's Inn
London WC1R 5JJ
London WC1R 5JJ (GB)

   


(54) DI-FLUORO CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS