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<ep-patent-document id="EP09718483B8W1" file="EP09718483W1B8.xml" lang="en" country="EP" doc-number="2262778" kind="B8" correction-code="W1" date-publ="20200101" status="c" dtd-version="ep-patent-document-v1-5">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCY..TRBGCZEEHUPLSK..HRIS..MTNO........................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 0.1.67 (18 Oct 2017) -  2999001/0</B007EP></eptags></B000><B100><B110>2262778</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20200101</date></B140><B150><B151>W1</B151><B153>54</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>09718483.2</B210><B220><date>20090305</date></B220><B240><B241><date>20100930</date></B241><B242><date>20140701</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>08425140</B310><B320><date>20080307</date></B320><B330><ctry>EP</ctry></B330></B300><B400><B405><date>20200101</date><bnum>202001</bnum></B405><B430><date>20101222</date><bnum>201051</bnum></B430><B450><date>20190821</date><bnum>201934</bnum></B450><B452EP><date>20190712</date></B452EP><B480><date>20200101</date><bnum>202001</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 231/54        20060101AFI20090929BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 401/12        20060101ALI20090929BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/416       20060101ALI20090929BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/435       20060101ALI20090929BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61P   3/10        20060101ALI20090929BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61P   9/00        20060101ALI20090929BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61P  13/00        20060101ALI20090929BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>1-BENZYL-3-HYDROXYMETHYLINDAZOLDERIVATE UND IHRE VERWENDUNG BEI DER BEHANDLUNG VON AUF DER EXPRESSION VON MCP-1, CX3CR1 UND P40 BASIERTEN ERKRANKUNGEN</B542><B541>en</B541><B542>1-BENZYL-3-HYDROXYMETHYLINDAZOLE DERIVATIVES AND USE THEREOF IN THE TREATMENT OF DISEASES BASED ON THE EXPRESSION OF MCP-1, CX3CR1 AND P40</B542><B541>fr</B541><B542>DÉRIVÉS DE 1-BENZYL-3-HYDROXYMÉTHYLINDAZOLE ET LEUR UTILISATION DANS LE TRAITEMENT DE MALADIES BASÉES SUR L'EXPRESSION DE MCP-1, CX3CR1 ET P40</B542></B540><B560><B561><text>WO-A-99/04770</text></B561><B561><text>WO-A1-2008/052898</text></B561><B561><text>CN-A- 101 074 208</text></B561><B561><text>US-A1- 2006 047 126</text></B561><B561><text>US-A1- 2007 043 057</text></B561><B562><text>HENKE B R ET AL: "Optimization of 3-(1H-indazol-3-ylmethyl)-1,5-benzodiazepi nes as potent, orally active CCK-A agonists" JOURNAL OF MEDICINAL CHEMISTRY, US AMERICAN CHEMICAL SOCIETY. WASHINGTON, vol. 40, no. 17, 15 August 1997 (1997-08-15), pages 2706-2725, XP002105882 ISSN: 0022-2623 cited in the application</text></B562><B562><text>CORSI, G. ET AL.: "1-halobenzyl-1H-indazoles-3-carboxylic acids. A new class of antispermatogenic agents" JOURNAL OF MEDICINAL CHEMISTRY, vol. 19, no. 6, 1976, pages 778-783, XP002493577 cited in the application</text></B562></B560></B500><B700><B720><B721><snm>GUGLIELMOTTI, Angelo</snm><adr><str>Via Gaetano Fuggetta 59</str><city>00149 Roma</city><ctry>IT</ctry></adr></B721><B721><snm>FURLOTTI, Guido</snm><adr><str>Via Ferdinando Palasciano 96</str><city>00151 Roma</city><ctry>IT</ctry></adr></B721><B721><snm>MANGANO, Giorgina</snm><adr><str>Via Gran Paradiso 84</str><city>00139 Roma</city><ctry>IT</ctry></adr></B721><B721><snm>CAZZOLLA, Nicola</snm><adr><str>Via Abetonia 20/L</str><city>00041 Albano Laziale (Roma)</city><ctry>IT</ctry></adr></B721></B720><B730><B731><snm>Aziende Chimiche Riunite Angelini 
Francesco A.C.R.A.F. S.p.A.</snm><iid>100082148</iid><irf>RA/08075/PCT/EP</irf><adr><str>Viale Amelia, 70</str><city>00181 Roma</city><ctry>IT</ctry></adr></B731></B730><B740><B741><snm>Colombo, Stefano Paolo</snm><sfx>et al</sfx><iid>101014935</iid><adr><str>Marchi &amp; Partners S.r.l. 
Via Vittor Pisani, 13</str><city>20124 Milano</city><ctry>IT</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MK</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>EP2009052588</anum></dnum><date>20090305</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2009109616</pnum></dnum><date>20090911</date><bnum>200937</bnum></B871></B870></B800></SDOBI>
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