(19)
(11) EP 2 265 615 A1

(12)

(43) Date of publication:
29.12.2010 Bulletin 2010/52

(21) Application number: 09721923.2

(22) Date of filing: 18.03.2009
(51) International Patent Classification (IPC): 
C07D 487/04(2006.01)
A61P 35/00(2006.01)
A61K 31/519(2006.01)
A61K 31/5025(2006.01)
 A61P 1/00(2006.01)
A61P 21/00(2006.01)
A61K 31/4985(2006.01)
(86) International application number:
PCT/EP2009/002012
(87) International publication number:
WO 2009/115321 (24.09.2009 Gazette 2009/39)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA RS

(30) Priority: 18.03.2008 EP 08005046
18.03.2008 US 37444

(71) Applicant: Santhera Pharmaceuticals (Schweiz) AG
4410 Liestal (CH)

(72) Inventors:
  • SOEBERDT, Michael
    79618 Rheinfelden (DE)
  • DEPPE, Holger
    CH-4052 Basel (CH)
  • ABEL, Ulrich
    69126 Heidelberg (DE)
  • FEURER, Achim
    79424 Auggen (DE)
  • METZ, Günther
    79541 Lörrach (DE)
  • OTT, Inge
    68775 Ketsch (DE)
  • HOFFMANN-ENGER, Barbara
    CH-4414 Füllinsdorf (CH)
  • NORDHOFF, Sonja
    CH-4144 Arlesheim (CH)

(74) Representative: Grünecker, Kinkeldey, Stockmair & Schwanhäusser Anwaltssozietät 
Leopoldstrasse 4
80802 München
80802 München (DE)

   


(54) IMIDAZOPYRIMIDINE, IMIDAZOPYRAZINE AND IMIDAZOPYRIDAZINE DERIVATIVES AS MELANOCORTIN-4 RECEPTOR MODULATORS