(19)
(11) EP 2 268 634 A2

(12)

(88) Date of publication A3:
05.11.2009

(43) Date of publication:
05.01.2011 Bulletin 2011/01

(21) Application number: 09718766.0

(22) Date of filing: 12.03.2009
(51) International Patent Classification (IPC): 
C07D 403/04(2006.01)
A61K 31/513(2006.01)
A61P 11/00(2006.01)
A61K 31/606(2006.01)
A61P 9/00(2006.01)
(86) International application number:
PCT/IB2009/005454
(87) International publication number:
WO 2009/112954 (17.09.2009 Gazette 2009/38)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA RS

(30) Priority: 13.03.2008 IN CH06282008

(71) Applicant: Actavis Group PTC EHF
220 Hafnarfjordur (IS)

(72) Inventors:
  • DIXIT, Girish
    Kaushambi Ghaziabad (up) 201010 (IN)
  • GAIKWAD, Nandkumar
    Maharashtra 410 210 (IN)
  • NAIDU, Hima, Prasad
    Andhra Pradesh (IN)
  • PRADHAN, Nitin, Sharadchandra
    Maharashtra 400601 (IN)
  • VALGEIRSSON, Jon
    IS-220 Hafnarfjorour (IS)

(74) Representative: Lasterra Sánchez, Elena 
HLBBshaw Merlin House Falconry Court Baker's Lane
GB-Epping, Essex CM16 5DQ
GB-Epping, Essex CM16 5DQ (GB)

   


(54) PROCESSES FOR THE PREPARATION OF BOSENTAN AND RELATED COMPOUNDS USING NOVEL INTERMEDIATES