(19)
(11) EP 2 276 748 A1

(12)

(43) Date of publication:
26.01.2011 Bulletin 2011/04

(21) Application number: 08742724.1

(22) Date of filing: 10.04.2008
(51) International Patent Classification (IPC): 
C07D 241/44(2006.01)
C07D 471/04(2006.01)
A61K 31/4985(2006.01)
 C07D 401/12(2006.01)
A61K 31/498(2006.01)
A61P 35/00(2006.01)
(86) International application number:
PCT/US2008/004631
(87) International publication number:
WO 2009/126123 (15.10.2009 Gazette 2009/42)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA MK RS

(71) Applicant: Gilead Sciences, Inc.
Foster City, CA 94404 (US)

(72) Inventors:
  • KOLTUN, Dmitry
    Foster City CA 94404 (US)
  • ZABLOCKI, Jeff
    San Mateo CA 94401 (US)
  • PARKHILL, Eric
    San Francisco CA 94122 (US)
  • GLUSHKOV, Andrei
    Moscow 117574 (RU)
  • VASILEVICH, Natalya
    Moscow 123480 (RU)
  • ZILBERSHTEIN, Timur
    Tomsk (RU)
  • IVANOV, Alexey
    Moscow 123367 (RU)
  • CHISHOLM, Jeffrey
    Mountain View CA 94040 (US)

(74) Representative: Reitstötter - Kinzebach 
Patentanwälte Sternwartstrasse 4
81679 München
81679 München (DE)

   


(54) BICYCLIC NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS FOR USE AS STEAROYL COA DESATURASE INHIBITORS