(19)
(11) EP 2 279 180 A1

(12)

(43) Date of publication:
02.02.2011 Bulletin 2011/05

(21) Application number: 09733825.5

(22) Date of filing: 23.04.2009
(51) International Patent Classification (IPC): 
C07D 261/20(2006.01)
A61P 25/00(2006.01)
A61K 31/423(2006.01)
(86) International application number:
PCT/EP2009/054859
(87) International publication number:
WO 2009/130263 (29.10.2009 Gazette 2009/44)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA RS

(30) Priority: 24.04.2008 IT MI20080768

(71) Applicant: Abiogen Pharma S.p.A.
56014 Ospedaletto (PI) (IT)

(72) Inventors:
  • NEGGIANI, Fabio
    I-56123 Pisa (IT)
  • NAPOLITANO, Elio
    I-56127 Pisa (IT)
  • BASAGNI, Simone
    I-56124 Pisa (IT)
  • POLITI, Barbara
    I-57124 Livorno (IT)

(74) Representative: Cattaneo, Elisabetta et al
Notarbartolo & Gervasi S.p.A. Corso di Porta Vittoria, 9
IT-20122 Milano
IT-20122 Milano (IT)

   


(54) PROCESS FOR PREPARING A CRYSTALLINE FORM COMPOUND OF 3-BENZYL-2-METHYL-2,3,3a,4,5,6,7,7a-OCTAHYDROBENZOÝd¨ISOXAZOL-4-ONE