(19)
(11) EP 2 280 951 A2

(12)

(88) Date of publication A3:
21.01.2010

(43) Date of publication:
09.02.2011 Bulletin 2011/06

(21) Application number: 08732845.6

(22) Date of filing: 26.03.2008
(51) International Patent Classification (IPC): 
C07D 319/20(2006.01)
A61P 25/08(2006.01)
 A61K 31/357(2006.01)
(86) International application number:
PCT/US2008/058247
(87) International publication number:
WO 2009/120192 (01.10.2009 Gazette 2009/40)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA MK RS

(71) Applicant: Janssen Pharmaceutica, N.V.
2340 Beerse (BE)

(72) Inventors:
  • BALLENTINE, Scott, A.
    Lansdale, Pennsylvania 19446 (US)
  • REANY, Laura
    Quakertown, PA 18951 (US)

(74) Representative: Warner, James Alexander 
Carpmaels & Ransford One Southampton Row
London WC1B 5HA
London WC1B 5HA (GB)

   


(54) PROCESSES FOR THE PREPARATION OF BENZO-FUSED DIOXIN DERIVATIVES