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<ep-patent-document id="EP09751280B8W1" file="EP09751280W1B8.xml" lang="en" country="EP" doc-number="2283020" kind="B8" correction-code="W1" date-publ="20121212" status="c" dtd-version="ep-patent-document-v1-4">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCY..TRBGCZEEHUPLSK..HRIS..MTNO........................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>DIM360 Ver 2.15 (14 Jul 2008) -  2999001/0</B007EP></eptags></B000><B100><B110>2283020</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20121212</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>09751280.0</B210><B220><date>20090518</date></B220><B240><B241><date>20101217</date></B241><B242><date>20110907</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>54345 P</B310><B320><date>20080519</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20121212</date><bnum>201250</bnum></B405><B430><date>20110216</date><bnum>201107</bnum></B430><B450><date>20121031</date><bnum>201244</bnum></B450><B452EP><date>20120515</date></B452EP><B480><date>20121212</date><bnum>201250</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 487/04        20060101AFI20091211BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/519       20060101ALI20091211BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61P  35/00        20060101ALI20091211BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>SUBSTITUIERTE IMIDAZOPYR- UND IMIDAZOTRIAZINE</B542><B541>en</B541><B542>SUBSTITUTED IMIDAZOPYR-AND IMIDAZOTRI-AZINES</B542><B541>fr</B541><B542>IMIDAZOPYRAZINES ET IMIDAZOTRIAZINES SUBSTITUÉES</B542></B540><B560><B561><text>WO-A-2006/004703</text></B561><B561><text>WO-A-2007/075554</text></B561><B561><text>US-A1- 2006 046 977</text></B561><B562><text>MULVIHILL ET AL: "Novel 2-phenylquinolin-7-yl-derived imidazo[1,5-a]pyrazines as potent insulin-like growth factor-I receptor (IGF-IR) inhibitors" BIOORGANIC &amp; MEDICINAL CHEMISTRY, ELSEVIER SCIENCE LTD, GB, vol. 16, no. 3, 23 October 2007 (2007-10-23), pages 1359-1375, XP022453107 ISSN: 0968-0896</text></B562><B562><text>KOPECKY D J ET AL: "Identification and optimization of N&lt;3&gt;,N&lt;6&gt;-diaryl-1H-pyrazolo[3,4-d ]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors" BIOORGANIC &amp; MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, vol. 18, no. 24, 15 December 2008 (2008-12-15), pages 6352-6356, XP025679027 ISSN: 0960-894X [retrieved on 2008-11-01]</text></B562></B560></B500><B700><B720><B721><snm>CREW, Andrew, P.</snm><adr><str>OSI Pharmaceuticals Inc.
Broadhollow Bioscience Park
1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B721><B721><snm>JIN, Meizhong</snm><adr><str>OSI Pharmaceuticals Inc.
Broadhollow Bioscience Park
1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B721><B721><snm>KADALBAJOO, Mridula</snm><adr><str>OSI Pharmaceuticals Inc.
Broadhollow Bioscience Park
1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B721><B721><snm>KLEINBERG, Andrew</snm><adr><str>OSI Pharmaceuticals Inc.
Broadhollow Bioscience Park
1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B721><B721><snm>MULVIHILL, Mark, J.</snm><adr><str>OSI Pharmaceuticals Inc.
Broadhollow Bioscience Park
1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B721><B721><snm>WANG, Jing</snm><adr><str>OSI Pharmaceuticals Inc.
Broadhollow Bioscience Park
1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>OSI Pharmaceuticals, LLC</snm><iid>101256668</iid><irf>42021-596N01EP</irf><adr><str>1 Bioscience Park Drive</str><city>Farmingdale, NY 11735</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Haile, Alison Victoria</snm><sfx>et al</sfx><iid>101087163</iid><adr><str>Mintz Levin, Cohn, Ferris, Glovsky and 
Popeo IP, LLP 
Alder Castle 
10 Noble Street</str><city>London EC2V 7JX</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MK</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>US2009044325</anum></dnum><date>20090518</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2009143051</pnum></dnum><date>20091126</date><bnum>200948</bnum></B871></B870><B880><date>20110216</date><bnum>201107</bnum></B880></B800></SDOBI>
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