(19)
(11) EP 2 285 376 A1

(12)

(43) Date of publication:
23.02.2011 Bulletin 2011/08

(21) Application number: 09747249.2

(22) Date of filing: 08.05.2009
(51) International Patent Classification (IPC): 
A61K 31/44(2006.01)
C07D 405/00(2006.01)
C07D 401/00(2006.01)
(86) International application number:
PCT/US2009/043302
(87) International publication number:
WO 2009/140164 (19.11.2009 Gazette 2009/47)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated Extension States:
AL BA RS

(30) Priority: 16.05.2008 US 53795

(71) Applicant: Chipscreen Biosciences Ltd.
Shenzhen 518057 (CN)

(72) Inventors:
  • LU, Xian-Ping
    Belle Meade NJ 08502 (US)
  • LI, Zhi-Bin
    Shenzhen 518057 (CN)
  • ZHI-QIANG, Ning
    Shenzhen 518057 (CN)

(74) Representative: Gowshall, Jonathan Vallance 
Forrester & Boehmert Pettenkoferstrasse 20-22
80336 München
80336 München (DE)

   


(54) 6-AMINONICOTINAMIDE DERIVATIVES AS POTENT AND SELECTIVE HISTONE DEACETYLASE INHIBITORS