TETRAHYDRO-PYRAZOLO[1,5-A]PYRIDO-PYRIMIDINES AS ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, METHODS FOR THE PRODUCTION AND USE THEREOF

(19)

(11)

EP 2 305 678 B8

(12)	CORRECTED EUROPEAN PATENT SPECIFICATION
	Note: Bibliography reflects the latest situation

(15)	Correction information:
	Corrected version no 1 (W1 B1)

(48)	Corrigendum issued on:
	05.03.2014 Bulletin 2014/10

(45)	Mention of the grant of the patent:
	25.12.2013 Bulletin 2013/52

(21)	Application number: 09742911.2

(22)	Date of filing: 30.04.2009

(51)

International Patent Classification (IPC):

C07D 471/14^(2006.01)
A61K 31/519^(2006.01)
A61P 25/18^(2006.01)
A61P 25/08^(2006.01)
A61P 25/26^(2006.01)
A61P 25/16^(2006.01)

A61P 25/22^(2006.01)
A61P 25/24^(2006.01)
A61P 25/28^(2006.01)
A61P 3/08^(2006.01)
A61P 9/10^(2006.01)
A61P 3/04^(2006.01)

(86)	International application number:
	PCT/RU2009/000209

(87)	International publication number:
	WO 2009/136814 (12.11.2009 Gazette 2009/46)

(54)

TETRAHYDRO-PYRAZOLO[1,5-A]PYRIDO-PYRIMIDINES AS ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, METHODS FOR THE PRODUCTION AND USE THEREOF

TETRAHYDROPYRAZOLO[1,5-A]PYRIDOPYRIMIDINE ALS ANTAGONISTEN VON SEROTONIN-5-HT6-REZEPTOREN, VERFAHREN ZU DEREN HERSTELLUNG UND DEREN VERWENDUNG

TETRAHYDRO-PYRAZOLOÝ1,5-A¨PYRIDO -PYRIMIDINES AGISSANT COMME DES ANTAGONISTES DES RÉCEPTEURS 5-HT6 DE SÉROTONINE ET PROCÉDÉS DE PRODUCTION ET D'UTILISATION CORRESPONDANTS

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR

(30)

Priority:

07.05.2008 RU 2008117845

(43)	Date of publication of application:
	06.04.2011 Bulletin 2011/14

(73)	Proprietors:
	Ivashchenko, Andrey Alexandrovich Moscow, 127576 (RU) Alla Chem, LLC. Carson City, NV 89701 (US)

(72)	Inventors:
	KYSIL, Volodymyr Mikhailovich Kiev 021140 (UA) SAVCHUK, Nikolay Filippovich Moscow 117420 (RU) IVASHCHENKO, Alexander Vasilievich Encinitas CA 92024 (US) IVASHCHENKO, Andrey Alexandrovich Moskow, 127576 (RU)

(74)	Representative: Henrion, Oliver et al
	Patentanwälte Zellentin & Partner Rubensstraße 30 DE-67061 Ludwigshafen DE-67061 Ludwigshafen (DE)

(56)

References cited: :

WO-A1-2007/147883
US-A- 4 066 645

US-A- 4 066 643
US-A- 4 072 680


	Remarks:
	The file contains technical information submitted after the application was filed and not included in this specification

Note: Within nine months from the publication of the mention of the grant of the European patent, any person may give notice to the European Patent Office of opposition to the European patent granted. Notice of opposition shall be filed in a written reasoned statement. It shall not be deemed to have been filed until the opposition fee has been paid. (Art. 99(1) European Patent Convention).