(19)
(11) EP 2 310 387 A2

(12)

(88) Date of publication A3:
05.08.2010

(43) Date of publication:
20.04.2011 Bulletin 2011/16

(21) Application number: 09777523.3

(22) Date of filing: 29.07.2009
(51) International Patent Classification (IPC): 
C07D 453/02(2006.01)
A61K 31/439(2006.01)
 A61P 13/10(2006.01)
(86) International application number:
PCT/EP2009/005497
(87) International publication number:
WO 2010/012459 (04.02.2010 Gazette 2010/05)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR
Designated Extension States:
AL BA RS

(30) Priority: 29.07.2008 SI 200800188
20.11.2008 SI 200800285
21.04.2009 SI 200900113

(71) Applicant: KRKA, D.D., Novo Mesto
8501 Novo mesto (SI)

(72) Inventors:
  • RU I , Milo
    SI-3000 Celje (SI)
  • PRUDI , Darja
    SI-8000 Novo Mesto (SI)
  • PE AVAR, Anica
    SI-8000 Novo Mesto (SI)
  • ZANOTTI-GEROSA, Antonio
    Cambridge CB1 2PY (GB)
  • STROPNIK, Tadej
    SI-1000 Ljublijana (SI)

(74) Representative: Westendorp | Sommer 
Uhlandstraße 2
80336 München
80336 München (DE)

   


(54) A PROCESS FOR THE PREPARATION OF SOLIFENACIN SALTS AND THEIR INCLUSION INTO PHARMACEUTICAL DOSAGE FORMS