(19)
(11) EP 2 344 463 A2

(12)

(88) Date of publication A3:
01.07.2010

(43) Date of publication:
20.07.2011 Bulletin 2011/29

(21) Application number: 09752053.0

(22) Date of filing: 04.11.2009
(51) International Patent Classification (IPC): 
C07D 275/02(2006.01)
C07D 417/04(2006.01)
C07D 417/12(2006.01)
C07D 513/10(2006.01)
A61P 9/00(2006.01)
A61P 25/00(2006.01)
A61P 35/00(2006.01)
C07D 275/04(2006.01)
C07D 417/06(2006.01)
C07D 513/04(2006.01)
A61K 31/425(2006.01)
A61P 11/00(2006.01)
A61P 29/00(2006.01)
A61P 37/00(2006.01)
(86) International application number:
PCT/US2009/063318
(87) International publication number:
WO 2010/054024 (14.05.2010 Gazette 2010/19)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR
Designated Extension States:
AL BA RS

(30) Priority: 04.11.2008 US 111041 P

(71) Applicant: Abbott Laboratories
Abbott Park, Illinois 60064-6008 (US)

(72) Inventors:
  • CARROLL, William, A.
    Evanston IL 60201 (US)
  • KOLASA, Teodozyj
    Lake Villa IL 60046 (US)
  • LI, Tongmei
    Lake Bluff IL 60044 (US)
  • NELSON, Derek, W.
    Highland Park IL 60035 (US)
  • PATEL, Meena, V.
    Green Oaks IL 60048 (US)
  • PEDDI, Sridhar
    Grayslake IL 60030 (US)
  • PEREZ-MEDRANO, Arturo
    Grayslake IL 60030 (US)
  • WANG, Xuequing
    Evanston IL 60202 (US)

(74) Representative: Modiano, Micaela Nadia et al
Modiano & Partners Thierschstrasse 11
80538 München
80538 München (DE)

   


(54) 1,2 -THIAZOL YL DERIVATIVES AS CANNABINOID RECEPTOR LIGANDS