(19)
(11) EP 2 350 029 A1

(12)

(43) Date of publication:
03.08.2011 Bulletin 2011/31

(21) Application number: 08825468.5

(22) Date of filing: 15.10.2008
(51) International Patent Classification (IPC): 
C07D 239/91(2006.01)
A61K 31/517(2006.01)
 C07D 471/04(2006.01)
A61P 3/00(2006.01)
(86) International application number:
PCT/US2008/079975
(87) International publication number:
WO 2010/056230 (20.05.2010 Gazette 2010/20)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR

(71) Applicant: Gilead Sciences, Inc.
Foster City, CA 94404 (US)

(72) Inventors:
  • KOLTUN, Dmitry
    Foster City CA 94404 (US)
  • PARKHILL, Eric
    San Francisco CA 94122 (US)
  • BOZE, Melanie
    Round Rock TX 78681 (US)
  • ZABLOCKI, Jeff
    Los Altos CA 94024 (US)
  • VASILEVICH, Natalya
    Moscow 123480 (RU)
  • MAYBORODA, Elena
    Mytishi 141014  (RU)
  • GLUSHKOV, Andrey
    Moscow 117574 (RU)
  • COLE, Andrew
    Robbinsville NJ 08691 (US)
  • CHISHOLM, Jeffrey
    Mountain View CA 94040 (US)

(74) Representative: Schnappauf, Georg et al
Dr. Volker Vossius Patent- und Rechtsanwaltskanzlei Geibelstrasse 6
81679 München
81679 München (DE)

   


(54) 3-HYDROQUINAZOLIN-4-ONE DERIVATIVES FOR USE AS STEAROYL COA DESATURASE INHIBITORS