(19)
(11) EP 2 362 874 A2

(12)

(88) Date of publication A3:
11.11.2010

(43) Date of publication:
07.09.2011 Bulletin 2011/36

(21) Application number: 09795592.6

(22) Date of filing: 06.11.2009
(51) International Patent Classification (IPC): 
C07D 405/12(2006.01)
(86) International application number:
PCT/US2009/063475
(87) International publication number:
WO 2010/054138 (14.05.2010 Gazette 2010/19)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR
Designated Extension States:
AL BA RS

(30) Priority: 06.11.2008 US 112152 P

(71) Applicant: Vertex Pharmaceuticals Incorporated
Cambridge, MA 02139 (US)

(72) Inventors:
  • RUAH, Sara S., Hadida
    La Jolla CA 92037 (US)
  • GROOTENHUIS, Peter, D.j.
    San Diego CA 92130 (US)
  • MILLER, Mark, T.
    San Diego CA 92109 (US)
  • MCCARTNEY, Jason
    Cardiff By The Sea CA 92007 (US)
  • VAN GOOR, Fredrick
    San Diego CA 92109 (US)
  • NUMA, Mehdi Michel, Djamel
    San Diego CA 92117 (US)
  • ZHOU, Jinglan
    San Diego CA 92130 (US)
  • BEAR, Brian
    Oceanside CA 92057 (US)

(74) Representative: Cohausz & Florack 
Bleichstraße 14
40211 Düsseldorf
40211 Düsseldorf (DE)

   


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