(19)
(11) EP 2 403 852 B8

(12) CORRECTED EUROPEAN PATENT SPECIFICATION
Note: Bibliography reflects the latest situation

(15) Correction information:
Corrected version no 1 (W1 B1)

(48) Corrigendum issued on:
17.12.2014 Bulletin 2014/51

(45) Mention of the grant of the patent:
29.10.2014 Bulletin 2014/44

(21) Application number: 10706659.9

(22) Date of filing: 05.03.2010
(51) International Patent Classification (IPC): 
C07D 235/30(2006.01)
C07D 405/12(2006.01)
C07D 403/12(2006.01)
 C07D 401/12(2006.01)
C07D 409/12(2006.01)
(86) International application number:
PCT/EP2010/052799
(87) International publication number:
WO 2010/100249 (10.09.2010 Gazette 2010/36)

(54)

2-AMINOBENZIMIDAZOLE-5-CARBOXAMIDES AS ANTI-INFLAMMATORY AGENTS

2-AMINOBENZIMIDAZOL-5-CARBONSÄUREAMIDE ALS ENTZÜNDUNGSHEMMENDE MITTEL

2-AMINOBENZIMIDAZOLE-5-CARBOXAMIDES EN TANT QU'ANTI-INFLAMMATOIRES

(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR
Designated Extension States:
AL BA ME RS

(30) Priority: 05.03.2009 EP 09154414
17.12.2009 EP 09179618

(43) Date of publication of application:
11.01.2012 Bulletin 2012/02

(73) Proprietor: Orexo AB
751 05 Uppsala (SE)

(72) Inventors:
  • PFAU, Roland
    55216 Ingelheim Am Rhein (DE)
  • ARNDT, Kirsten
    55216 Ingelheim Am Rhein (DE)
  • DOODS, Henri
    55216 Ingelheim Am Rhein (DE)
  • KLINDER, Klaus
    55216 Ingelheim Am Rhein (DE)
  • KUELZER, Raimund
    55216 Ingelheim Am Rhein (DE)
  • LUBRIKS, Dimitrijs
    1006 Riga (LV)
  • MACK, Juergen
    55216 Ingelheim Am Rhein (DE)
  • PELCMAN, Benjamin
    75105 Uppsala (SE)
  • PRIEPKE, Henning
    55216 Ingelheim Am Rhein (DE)
  • ROENN, Robert
    75105 Uppsala (SE)
  • STENKAMP, Dirk
    55216 Ingelheim Am Rhein (DE)
  • SUNA, Edgars
    1006 Riga (LV)

(74) Representative: Potter Clarkson LLP 
The Belgrave Centre Talbot Street
Nottingham, NG1 5GG
Nottingham, NG1 5GG (GB)


(56) References cited: : 
WO-A-00/49005
WO-A-00/68213
WO-A-03/053939
WO-A-2005/070920
WO-A-2007/095124
WO-A1-2010/034796
WO-A1-2010/034798
WO-A2-2008/009924
FR-A- 2 852 957
US-A1- 2007 060 598
 WO-A-00/61580
WO-A-01/25238
WO-A-2005/070906
WO-A-2006/077366
WO-A1-2008/071944
WO-A1-2010/034797
WO-A1-2010/034799
FR-A- 2 851 563
US-A1- 2006 287 344
   
  • R. D. CARPENTER ET AL.: "Carbodiimide-based benzimidazole library method" JOURNAL OF COMBINATORIAL CHEMISTRY, vol. 8, no. 6, 27 October 2006 (2006-10-27), pages 907-914, XP002557183
   
Note: Within nine months from the publication of the mention of the grant of the European patent, any person may give notice to the European Patent Office of opposition to the European patent granted. Notice of opposition shall be filed in a written reasoned statement. It shall not be deemed to have been filed until the opposition fee has been paid. (Art. 99(1) European Patent Convention).