(19)
(11) EP 2 406 271 A1

(12)

(43) Date of publication:
18.01.2012 Bulletin 2012/03

(21) Application number: 09764844.8

(22) Date of filing: 07.12.2009
(51) International Patent Classification (IPC): 
C07H 17/02(2006.01)
 A61K 31/7056(2006.01)
(86) International application number:
PCT/EP2009/066551
(87) International publication number:
WO 2010/066690 (17.06.2010 Gazette 2010/24)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR
Designated Extension States:
AL BA RS

(30) Priority: 08.12.2008 EP 08291157

(71) Applicant: SANOFI
75013 Paris (FR)

(72) Inventors:
  • BERCHTOLD, Harald
    65926 Frankfurt am Main (DE)
  • NAGEL, Norbert
    65926 Frankfurt am Main (DE)
  • BAUMGARTNER, Bruno
    65926 Frankfurt am Main (DE)
  • PLETTENBURG, Oliver
    65926 Frankfurt am Main (DE)
  • WEIBERTH, Franz
    New Jersey 08807 (US)
  • HARPAL, Gill
    New Jersey 08807 (US)
  • YU, Yong
    New Jersey 08807 (US)
  • LIEBERMAN, Harvey
    New Jersey 08807 (US)
  • SECORD, Elisabeth
    New Jersey 08807 (US)
  • GORDONOV, Boris
    New Jersey 08807 (US)
  • DONEGHAN, Tim
    New Jersey 08807 (US)
  • BYARD, Steve
    New Jersey 08807 (US)

(74) Representative: Fischer, Hans-Jürgen et al
Sanofi-Aventis Deutschland GmbH Patents Germany Industriepark Höchst Gebäude K 801
65926 Frankfurt am Main
65926 Frankfurt am Main (DE)

   


(54) A NOVEL CRYSTALLINE HETEROAROMATIC FLUOROGLYCOSIDE HYDRATE, PROCESSES FOR MAKING, METHODS OF USE AND PHARMACEUTICAL COMPOSITIONS THEREOF