(19)
(11) EP 2 414 351 A1

(12)

(43) Date of publication:
08.02.2012 Bulletin 2012/06

(21) Application number: 10714103.8

(22) Date of filing: 30.03.2010
(51) International Patent Classification (IPC): 
C07D 403/12(2006.01)
A61K 31/53(2006.01)
A61P 25/28(2006.01)
(86) International application number:
PCT/JP2010/056143
(87) International publication number:
WO 2010/114162 (07.10.2010 Gazette 2010/40)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR

(30) Priority: 31.03.2009 CA 2660954

(71) Applicant: Astellas Pharma Inc.
Tokyo 103-8411 (JP)

(72) Inventors:
  • OHMORI Junya
    Tokyo 1038411 (JP)
  • KASAI Makoto
    Tokyo 1038411 (JP)
  • KIMURA Takenori
    Tokyo 1038411 (JP)
  • HAMADA Noritaka
    Tokyo 1038411 (JP)
  • MIZOGUCHI Ryo
    Tokyo 1038411 (JP)
  • MIYAMOTO Satoshi
    Tokyo 1038411 (JP)
  • KAWANO Noriyuki
    Tokyo 1038411 (JP)

(74) Representative: HOFFMANN EITLE 
Patent- und Rechtsanwälte Arabellastraße 4
81925 München
81925 München (DE)

   


(54) NOVEL SALT OF 1,3,5-TRIAZINE-2,4,6-TRIAMINE DERIVATIVE