(19)
(11) EP 2 432 771 A1

(12)

(43) Date of publication:
28.03.2012 Bulletin 2012/13

(21) Application number: 10778279.9

(22) Date of filing: 18.05.2010
(51) International Patent Classification (IPC): 
C07D 261/02(2006.01)
(86) International application number:
PCT/US2010/035309
(87) International publication number:
WO 2010/135360 (25.11.2010 Gazette 2010/47)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR

(30) Priority: 18.05.2009 US 179285 P
18.05.2009 US 179280 P
18.05.2009 US 179283 P

(71) Applicant: Infinity Pharmaceuticals, Inc.
Cambridge, MA 02139 (US)

(72) Inventors:
  • BEHNKE, Mark, L.
    Somerville MA 02144 (US)
  • CASTRO, Alfredo, C.
    Winchester MA 01890 (US)
  • CHAN, Lawrence, K.
    Brookline MA 02446 (US)
  • EVANS, Catherine, A.
    Somerville MA 02145 (US)
  • GRENIER, Louis
    Newton MA 02458 (US)
  • GROGAN, Michael, J.
    Winchester MA 01890 (US)
  • LEBLANC, Yves
    Canada H9J 3Y3 (CA)
  • LIU, Tao
    Ashland MA 01721 (US)
  • PELUSO, Stephane
    Somerville MA 02144 (US)
  • SNYDER, Daniel, A.
    Somerville MA 02145 (US)
  • TIBBITTS, Thomas, T.
    Westford MA 01886 (US)

(74) Representative: Ritter, Thomas Kurt et al
Jones Day Prinzregentenstraße 11
80538 München
80538 München (DE)

   


(54) ISOXAZOLINES AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE