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<ep-patent-document id="EP10763963A1" file="10763963.5" lang="en" country="EP" doc-number="2486011" kind="A1" date-publ="20120815" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................</B001EP><B003EP>*</B003EP><B005EP>X</B005EP><B007EP>DIM360 Ver 2.15 (14 Jul 2008) -  1100000/0</B007EP></eptags></B000><B100><B110>2486011</B110><B130>A1</B130><B140><date>20120815</date></B140><B190>EP</B190></B100><B200><B210>10763963.5</B210><B220><date>20101006</date></B220><B240><B241><date>20120405</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>250229 P</B310><B320><date>20091009</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20120815</date><bnum>201233</bnum></B405><B430><date>20120815</date><bnum>201233</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 207/40        20060101AFI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 213/40        20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07D 231/12        20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07D 277/32        20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>C07C 233/05        20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61K  31/40        20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61K  31/415       20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>A61K  31/425       20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>A61K  31/4406      20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>A61P   3/00        20060101ALI20110427BHEP        </text></classification-ipcr><classification-ipcr sequence="11"><text>A61P  25/00        20060101ALI20110427BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>MODULATOREN DES G-PROTEIN-GEKOPPELTEN REZEPTORS 88</B542><B541>en</B541><B542>MODULATORS OF G PROTEIN-COUPLED RECEPTOR 88</B542><B541>fr</B541><B542>MODULATEURS DES RÉCEPTEURS COUPLÉS AUX PROTÉINES G 88</B542></B540></B500><B700><B710><B711><snm>Bristol-Myers Squibb Company</snm><iid>101100473</iid><irf>M/53095-EP</irf><adr><str>Route 206 and Provinceline Road 
P.O. Box 4000</str><city>Princeton NJ 08543-4000</city><ctry>US</ctry></adr></B711><B711><snm>Lexicon Pharmaceuticals, Inc.</snm><iid>100964378</iid><irf>M/53095-EP</irf><adr><str>8800 Technology Forest Place</str><city>The Woodlands, TX 77381</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>DZIERBA, Carolyn, Diane</snm><adr><str>c/o Bristol-Myers Squibb Company
5 Research Parkway</str><city>Wallingford, Connecticut 06492</city><ctry>US</ctry></adr></B721><B721><snm>HARTZ, Richard, A.</snm><adr><str>c/o Bristol-Myers Squibb Company
5 Research Parkway</str><city>Wallingford, Connecticut 06492</city><ctry>US</ctry></adr></B721><B721><snm>BI, Yingzhi</snm><adr><str>5 Mershon Lane</str><city>Plainsboro, New Jersey 08536</city><ctry>US</ctry></adr></B721><B721><snm>AHUJA, Vijay T.</snm><adr><str>c/o Bristol-Myers Squibb Company
5 Research Parkway</str><city>Wallingford, Connecticut 06492</city><ctry>US</ctry></adr></B721><B721><snm>BRONSON, Joanne J.</snm><adr><str>c/o Bristol-Myers Squibb Company
5 Research Parkway</str><city>Wallingford, Connecticut 06492</city><ctry>US</ctry></adr></B721><B721><snm>CARSON, Kenneth</snm><adr><str>96 Herrontown Road</str><city>Princeton, New Jersey 08540</city><ctry>US</ctry></adr></B721><B721><snm>CIANCHETTA, Giovanni</snm><adr><str>91 Gordon Avenue</str><city>Lawrenceville, New Jersey 08648</city><ctry>US</ctry></adr></B721><B721><snm>GREEN, Michael</snm><adr><str>1184 Dewalt Drive</str><city>Easton, Pennsylvania 18040</city><ctry>US</ctry></adr></B721><B721><snm>KIMBALL, David</snm><adr><str>13 Charred Oak Lane</str><city>East Windsor, New Jersey 08520</city><ctry>US</ctry></adr></B721><B721><snm>KIMURA, S. Roy</snm><adr><str>c/o Bristol-Myers Squibb Company
5 Research Parkway</str><city>Wallingford, Connecticut 06492</city><ctry>US</ctry></adr></B721><B721><snm>KWON, Soojin</snm><adr><str>70 Whitman Street</str><city>Haworth, New Jersey 07641</city><ctry>US</ctry></adr></B721><B721><snm>MACOR, John E.</snm><adr><str>c/o Bristol-Myers Squibb Company
5 Research Parkway</str><city>Wallingford, Connecticut 06492</city><ctry>US</ctry></adr></B721><B721><snm>ZHANG, Yulian</snm><adr><str>571 Aspen Woods Drive</str><city>Yardley, Pennsylvania 19067</city><ctry>US</ctry></adr></B721><B721><snm>ZIPP, Greg</snm><adr><str>52 Hillside Drive</str><city>Robbinsville, New Jersey 08691</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Reitstötter - Kinzebach</snm><iid>100061448</iid><adr><str>Patentanwälte 
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