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<ep-patent-document id="EP10799037B8W1" file="EP10799037W1B8.xml" lang="en" country="EP" doc-number="2516420" kind="B8" correction-code="W1" date-publ="20181017" status="c" dtd-version="ep-patent-document-v1-5">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 0.1.63 (23 May 2017) -  2999001/0</B007EP></eptags></B000><B100><B110>2516420</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20181017</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>10799037.6</B210><B220><date>20101222</date></B220><B240><B241><date>20120621</date></B241><B242><date>20160104</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>09382302</B310><B320><date>20091223</date></B320><B330><ctry>EP</ctry></B330><B310>307579 P</B310><B320><date>20100224</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20181017</date><bnum>201842</bnum></B405><B430><date>20121031</date><bnum>201244</bnum></B430><B450><date>20180822</date><bnum>201834</bnum></B450><B452EP><date>20180409</date></B452EP><B480><date>20181017</date><bnum>201842</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 401/14        20060101AFI20110714BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 403/04        20060101ALI20110714BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07D 403/14        20060101ALI20110714BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07D 409/14        20060101ALI20110714BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/506       20060101ALI20110714BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61P  29/00        20060101ALI20110714BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61P  37/08        20060101ALI20110714BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>AMINOALKYLPYRIMIDIN-DERIVATE ALS HISTAMIN-H4-REZEPTOR-ANTAGONISTEN</B542><B541>en</B541><B542>AMINOALKYLPYRIMIDINE DERIVATIVES AS HISTAMINE H4 RECEPTOR ANTAGONISTS</B542><B541>fr</B541><B542>DÉRIVÉS D'AMINOALKYLPYRIMIDINE EN TANT QU'ANTAGONISTES DU RÉCEPTEUR H4 DE L'HISTAMINE</B542></B540><B560><B561><text>EP-A- 1 505 064</text></B561><B561><text>WO-A-2004/039796</text></B561><B561><text>WO-A-2009/068512</text></B561><B561><text>WO-A-2009/080721</text></B561><B561><text>WO-A1-2006/110763</text></B561><B562><text>COWART M D ET AL: "Rotationally Constrained 2,4-Diamino-5,6-disubstituted Pyrimidines: A New Class of Histamine H4 Receptor Antagonists with Improved Druglikeness and in Vivo Efficacy in Pain and Inflammation Models", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, US, vol. 51, 26 September 2008 (2008-09-26), pages 6547-6557, XP002543231, ISSN: 0022-2623 [retrieved on 2008-09-26]</text></B562></B560></B500><B700><B720><B721><snm>CARCELLER GONZÁLEZ, Elena</snm><adr><str>Joan Miró 2</str><city>E-08190 Sant Cugat del Vallès</city><ctry>ES</ctry></adr></B721><B721><snm>VIRGILI BERNADO, Marina</snm><adr><str>Plaza Lesseps 11</str><city>E-08023 Barcelona</city><ctry>ES</ctry></adr></B721><B721><snm>SOLIVA SOLIVA, Robert</snm><adr><str>Frederica Montseny 42-44 5° 4ª</str><city>E-08980 Sant Feliu de Llobregat</city><ctry>ES</ctry></adr></B721><B721><snm>FERRER COSTA, Carles</snm><adr><str>Indústria 84-86 2° 2ª</str><city>E-08370 Calella</city><ctry>ES</ctry></adr></B721></B720><B730><B731><snm>Medicis Pharmaceutical Corporation</snm><iid>101764231</iid><irf>156 645 aa/sis</irf><adr><str>400 Somerset Corporate Blvd.</str><city>Bridgewater, NJ 08807</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Hoffmann Eitle</snm><iid>100061036</iid><adr><str>Patent- und Rechtsanwälte PartmbB 
Arabellastraße 30</str><city>81925 München</city><ctry>DE</ctry></adr></B741></B740></B700><B800><B840><ctry>AL</ctry><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MK</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>RS</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>SM</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>EP2010070562</anum></dnum><date>20101222</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2011076878</pnum></dnum><date>20110630</date><bnum>201126</bnum></B871></B870></B800></SDOBI>
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