(19)
(11) EP 2 531 190 A1

(12)

(43) Date of publication:
12.12.2012 Bulletin 2012/50

(21) Application number: 11700964.7

(22) Date of filing: 28.01.2011
(51) International Patent Classification (IPC): 
A61K 31/351(2006.01)
A61K 31/439(2006.01)
A61K 31/4433(2006.01)
C07D 407/04(2006.01)
A61P 25/00(2006.01)
A61K 31/4025(2006.01)
A61K 31/4412(2006.01)
C07D 309/14(2006.01)
A61P 29/00(2006.01)
(86) International application number:
PCT/EP2011/051179
(87) International publication number:
WO 2011/095434 (11.08.2011 Gazette 2011/32)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

(30) Priority: 02.02.2010 EP 10152359

(71) Applicant: F.Hoffmann-La Roche AG
4070 Basel (CH)

(72) Inventors:
  • KOLCZEWSKI, Sabine
    79540 Loerrach (DE)
  • PINARD, Emmanuel
    F-68480 Linsdorf (FR)

(74) Representative: Poppe, Regina 
F.Hoffmann-La Roche AG Patent Department Grenzacherstrasse 124
4070 Basel
4070 Basel (CH)

   


(54) TETRAHYDRO-PYRAN DERIVATIVES AGAINST NEUROLOGICAL ILLNESSES