(19)
(11)
EP 2 531 190 A1
(12)
(43)
Date of publication:
12.12.2012
Bulletin 2012/50
(21)
Application number:
11700964.7
(22)
Date of filing:
28.01.2011
(51)
International Patent Classification (IPC):
A61K
31/351
(2006.01)
A61K
31/439
(2006.01)
A61K
31/4433
(2006.01)
C07D
407/04
(2006.01)
A61P
25/00
(2006.01)
A61K
31/4025
(2006.01)
A61K
31/4412
(2006.01)
C07D
309/14
(2006.01)
A61P
29/00
(2006.01)
(86)
International application number:
PCT/EP2011/051179
(87)
International publication number:
WO 2011/095434
(
11.08.2011
Gazette 2011/32)
(84)
Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
(30)
Priority:
02.02.2010
EP 10152359
(71)
Applicant:
F.Hoffmann-La Roche AG
4070 Basel (CH)
(72)
Inventors:
KOLCZEWSKI, Sabine
79540 Loerrach (DE)
PINARD, Emmanuel
F-68480 Linsdorf (FR)
(74)
Representative:
Poppe, Regina
F.Hoffmann-La Roche AG Patent Department Grenzacherstrasse 124
4070 Basel
4070 Basel (CH)
(54)
TETRAHYDRO-PYRAN DERIVATIVES AGAINST NEUROLOGICAL ILLNESSES