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<ep-patent-document id="EP11722429B8W1" file="EP11722429W1B8.xml" lang="en" country="EP" doc-number="2575898" kind="B8" correction-code="W1" date-publ="20210421" status="c" dtd-version="ep-patent-document-v1-5">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 1.7.2 (20 November 2019) -  2999001/0</B007EP><B070EP>The file contains technical information submitted after the application was filed and not included in this specification</B070EP></eptags></B000><B100><B110>2575898</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20210421</date></B140><B150><B151>W1</B151><B153>54</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>11722429.5</B210><B220><date>20110530</date></B220><B240><B241><date>20121228</date></B241><B242><date>20170720</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>10164948</B310><B320><date>20100604</date></B320><B330><ctry>EP</ctry></B330></B300><B400><B405><date>20210421</date><bnum>202116</bnum></B405><B430><date>20130410</date><bnum>201315</bnum></B430><B450><date>20200930</date><bnum>202040</bnum></B450><B452EP><date>20200420</date></B452EP><B472><B475><date>20200930</date><ctry>FI</ctry><date>20201231</date><ctry>GR</ctry><date>20200930</date><ctry>HR</ctry><date>20200930</date><ctry>LV</ctry><date>20201230</date><ctry>NO</ctry><date>20200930</date><ctry>RS</ctry><date>20201230</date><ctry>BG</ctry></B475></B472><B480><date>20210421</date><bnum>202116</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>A61K  51/04        20060101AFI20200220BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K 101/02        20060101ALI20200220BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07B  59/00        20060101ALI20200220BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07C 213/08        20060101ALI20200220BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>VERFAHREN ZUR HERSTELLUNG VON F-18-MARKIERTEN AMYLOID-BETA-LIGANDEN</B542><B541>en</B541><B542>METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGAND</B542><B541>fr</B541><B542>PROCÉDÉ DE PRODUCTION DE LIGAND DE L'AMYLOÏDE BÊTA MARQUÉ AU 18F</B542></B540><B560><B561><text>WO-A1-2010/078370</text></B561><B561><text>WO-A1-2011/003591</text></B561><B561><text>WO-A2-2010/000409</text></B561><B561><text>US-A1- 2006 269 473</text></B561><B561><text>US-A1- 2010 113 763</text></B561><B562><text>ZHANG ET AL: "F-18 Polyethyleneglycol stilbenes as PET imaging agents targeting Abeta aggregates in the brain", NUCLEAR MEDICINE AND BIOLOGY, ELSEVIER, NY, US, vol. 32, no. 8, 1 November 2005 (2005-11-01), pages 799-809, XP005129336, ISSN: 0969-8051, DOI: 10.1016/J.NUCMEDBIO.2005.06.001 cited in the application</text></B562><B562><text>WANG H ET AL: "Facile and rapid one-step radiosynthesis of [&lt;18&gt;F]BAY94-9172 with a new precursor", NUCLEAR MEDICINE AND BIOLOGY, ELSEVIER, NY, US, vol. 38, no. 1, 1 January 2011 (2011-01-01), pages 121-127, XP027589497, ISSN: 0969-8051 [retrieved on 2010-08-16] cited in the application</text></B562><B562><text>PATT M ET AL: "Metabolite analysis of [18F]Florbetaben (BAY 94-9172) in human subjects: a substudy within a proof of mechanism clinical trial", JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY, KLUWER ACADEMIC PUBLISHERS, DO, vol. 284, no. 3, 16 March 2010 (2010-03-16), pages 557-562, XP019792449, ISSN: 1588-2780</text></B562><B562><text>LIN K J ET AL: "Whole-body biodistribution and brain PET imaging with [&lt;18&gt;F]AV-45, a novel amyloid imaging agent - a pilot study", NUCLEAR MEDICINE AND BIOLOGY, ELSEVIER, NY, US, vol. 37, no. 4, 1 May 2010 (2010-05-01), pages 497-508, XP027039103, ISSN: 0969-8051 [retrieved on 2010-04-07]</text></B562><B562><text>LIU Y ET AL: "Optimization of automated radiosynthesis of [&lt;18&gt;F]AV-45: a new PET imaging agent for Alzheimer's disease", NUCLEAR MEDICINE AND BIOLOGY, ELSEVIER, NY, US, vol. 37, no. 8, 1 November 2010 (2010-11-01), pages 917-925, XP027472064, ISSN: 0969-8051, DOI: 10.1016/J.NUCMEDBIO.2010.05.001 [retrieved on 2010-06-29] cited in the application</text></B562><B562><text>YAO C H ET AL: "GMP-compliant automated synthesis of [&lt;18&gt;F]AV-45 (Florbetapir F 18) for imaging beta-amyloid plaques in human brain", APPLIED RADIATION AND ISOTOPES, ELSEVIER, OXFORD, GB, vol. 68, no. 12, 1 December 2010 (2010-12-01), pages 2293-2297, XP027265706, ISSN: 0969-8043 [retrieved on 2010-07-07] cited in the application</text></B562><B562><text>PIYUSH KUMAR ET AL: "18F-FESB: synthesis and automated radiofluorination of a novel18F-labeled pet tracer for[beta]-amyloid plaques", JOURNAL OF LABELLED COMPOUNDS AND RADIOPHARMACEUTICALS, vol. 48, no. 13, 1 November 2005 (2005-11-01), pages 983-996, XP55006268, ISSN: 0362-4803, DOI: 10.1002/jlcr.1011</text></B562></B560></B500><B700><B720><B721><snm>BERNDT, Mathias</snm><adr><str>Lepsiusstr. 42</str><city>12163 Berlin</city><ctry>DE</ctry></adr></B721><B721><snm>FRIEBE, Matthias</snm><adr><str>Räuschstr. 8</str><city>13509 Berlin</city><ctry>DE</ctry></adr></B721><B721><snm>HULTSCH, Christina</snm><adr><str>Gontermannstr. 82</str><city>12101 Berlin</city><ctry>DE</ctry></adr></B721><B721><snm>SAMSON, Fabrice</snm><adr><str>301, 3rd Fl. Plus III
124-13 Itaewon-dong
Yongsan-gu</str><city>Seoul 140-858</city><ctry>KR</ctry></adr></B721><B721><snm>OH, Seung, Jun</snm><adr><str>205-501 Yowon 2nd Apt.
Yeongdeungpo-Gu</str><city>Seoul 150-045</city><ctry>KR</ctry></adr></B721><B721><snm>SMUDA, Christoph</snm><adr><str>Hangstr. 3</str><city>CH-8952 Schlieren</city><ctry>CH</ctry></adr></B721></B720><B730><B731><snm>Life Molecular Imaging SA</snm><iid>101782851</iid><irf>P75012EP01</irf><adr><str>Route de l'Ecole 13</str><city>1753 Matran</city><ctry>CH</ctry></adr></B731></B730><B740><B741><snm>Kilger, Ute</snm><iid>101135293</iid><adr><str>Boehmert &amp; Boehmert 
Anwaltspartnerschaft mbB 
Pettenkoferstrasse 22</str><city>80336 München</city><ctry>DE</ctry></adr></B741></B740></B700><B800><B840><ctry>AL</ctry><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MK</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>RS</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>SM</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>EP2011058819</anum></dnum><date>20110530</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2011151282</pnum></dnum><date>20111208</date><bnum>201149</bnum></B871></B870></B800></SDOBI>
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